网站主页 >> CAS数据库列表 >> H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
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- CAS号:
- 434938-41-7
- 英文名:
- K 41498
- 英文别名:
- K 41498;M.W. 3630.07 C162H276N48O46;D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
- 中文名:
- H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
- 中文别名:
- CRF2受体拮抗剂多肽;K41498 TFA 盐;H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
- CBNumber:
- CB8356040
- 分子式:
- C162H276N48O46
- 分子量:
- 3632.22
- MOL File:
- 434938-41-7.mol
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H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2化学性质
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储存条件:
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−20°C
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溶解度:
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Water (Slightly)
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形态:
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solid
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颜色:
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off-white
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水溶解性:
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Soluble to 5 mg/ml in water
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H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2性质、用途与生产工艺
K41498 是一种强选择性的 CRF2 receptor 拮抗剂,其对人 CRF2α、CRF2β 和 CRF1 受体的 Ki 值分别为 0.66 nM、0.62 nM 和 425 nM。K41498 是 antisauvagine-30 (aSvg-30) 的类似物,可抑制 sauvagine 刺激的 cAMP 在 hCRF2α/hCRF2β 表达细胞中的积累。K41498 可用于低血压研究。
H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
上下游产品信息
上游原料
下游产品
H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
生产厂家
434938-41-7, H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2 相关搜索:
- Releasing Factors
- Neuropeptides
- CRF
- CRF receptor and related
- 药靶配体
- 目录肽
- C162H276N48O46
- K41498 TFA 盐
- CRF2受体拮抗剂多肽
- H-D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
- 434938-41-7
- D-PHE-HIS-LEU-LEU-ARG-LYS-NLE-ILE-GLU-ILE-GLU-LYS-GLN-GLU-LYS-GLU-LYS-GLN-GLN-ALA-ALA-ASN-ASN-ARG-LEU-LEU-LEU-ASP-THR-ILE-NH2
- K 41498
- M.W. 3630.07 C162H276N48O46