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ChemicalBook >> CAS DataBase List >> Relugolix

Relugolix

Relugolix price.
  • $32 - $3728.1
  • Product name: Relugolix
  • CAS: 737789-87-6
  • MF: C29H27F2N7O5S
  • MW: 623.63
  • EINECS:237-099-7
  • MDL Number:MFCD25976856
  • Synonyms:TAK-385;TKA-385 Relugolix;TAK-385,Relugolix;CS-2851;TAK-385;TAK 385;TAK385;1-[4-[1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-3-methoxyurea;10G,100G,500G,1KG;N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxy urea
20 prices
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Brand
  • AK Scientific
  • Biorbyt Ltd
  • Cayman Chemical
  • ChemScene
  • Crysdot
  • DC Chemicals
Package
  • 1mg
  • 5mg
  • 10mg
  • 25mg
  • 50mg
  • 100mg
  • 250mg
  • 1g
  • ManufacturerAK Scientific
  • Product number6863CR
  • Product descriptionRelugolix
  • Packaging10mg
  • Price$370
  • Updated2021-12-16
  • Buy
  • ManufacturerAK Scientific
  • Product number6863CR
  • Product descriptionRelugolix
  • Packaging25mg
  • Price$691
  • Updated2021-12-16
  • Buy
  • ManufacturerBiorbyt Ltd
  • Product numberorb573025
  • Product descriptionRelugolix (TAK-385) >98%
  • Packaging100mg
  • Price$1133.9
  • Updated2021-12-16
  • Buy
  • ManufacturerBiorbyt Ltd
  • Product numberorb573025
  • Product descriptionRelugolix (TAK-385) >98%
  • Packaging250mg
  • Price$1802
  • Updated2021-12-16
  • Buy
  • ManufacturerBiorbyt Ltd
  • Product numberorb573025
  • Product descriptionRelugolix (TAK-385) >98%
  • Packaging1g
  • Price$3728.1
  • Updated2021-12-16
  • Buy
  • ManufacturerCayman Chemical
  • Product number29512
  • Product descriptionTAK-385
  • Packaging1mg
  • Price$32
  • Updated2024-03-01
  • Buy
  • ManufacturerCayman Chemical
  • Product number29512
  • Product descriptionTAK-385
  • Packaging5mg
  • Price$139
  • Updated2024-03-01
  • Buy
  • ManufacturerCayman Chemical
  • Product number29512
  • Product descriptionTAK-385
  • Packaging10mg
  • Price$243
  • Updated2024-03-01
  • Buy
  • ManufacturerCayman Chemical
  • Product number29512
  • Product descriptionTAK-385
  • Packaging25mg
  • Price$533
  • Updated2024-03-01
  • Buy
  • ManufacturerChemScene
  • Product numberCS-5917
  • Product descriptionRelugolix >98.0%
  • Packaging1mg
  • Price$70
  • Updated2021-12-16
  • Buy
  • ManufacturerChemScene
  • Product numberCS-5917
  • Product descriptionRelugolix >98.0%
  • Packaging5mg
  • Price$120
  • Updated2021-12-16
  • Buy
  • ManufacturerChemScene
  • Product numberCS-5917
  • Product descriptionRelugolix >98.0%
  • Packaging10mg
  • Price$190
  • Updated2021-12-16
  • Buy
  • ManufacturerChemScene
  • Product numberCS-5917
  • Product descriptionRelugolix >98.0%
  • Packaging50mg
  • Price$660
  • Updated2021-12-16
  • Buy
  • ManufacturerChemScene
  • Product numberCS-5917
  • Product descriptionRelugolix >98.0%
  • Packaging100mg
  • Price$1100
  • Updated2021-12-16
  • Buy
  • ManufacturerCrysdot
  • Product numberCD11064717
  • Product descriptionRelugolix(TAK385) 97%
  • Packaging5mg
  • Price$245
  • Updated2021-12-16
  • Buy
  • ManufacturerCrysdot
  • Product numberCD11064717
  • Product descriptionRelugolix(TAK385) 97%
  • Packaging10mg
  • Price$350
  • Updated2021-12-16
  • Buy
Manufacturer Product number Product description Packaging Price Updated Buy
AK Scientific 6863CR Relugolix 10mg $370 2021-12-16 Buy
AK Scientific 6863CR Relugolix 25mg $691 2021-12-16 Buy
Biorbyt Ltd orb573025 Relugolix (TAK-385) >98% 100mg $1133.9 2021-12-16 Buy
Biorbyt Ltd orb573025 Relugolix (TAK-385) >98% 250mg $1802 2021-12-16 Buy
Biorbyt Ltd orb573025 Relugolix (TAK-385) >98% 1g $3728.1 2021-12-16 Buy
Cayman Chemical 29512 TAK-385 1mg $32 2024-03-01 Buy
Cayman Chemical 29512 TAK-385 5mg $139 2024-03-01 Buy
Cayman Chemical 29512 TAK-385 10mg $243 2024-03-01 Buy
Cayman Chemical 29512 TAK-385 25mg $533 2024-03-01 Buy
ChemScene CS-5917 Relugolix >98.0% 1mg $70 2021-12-16 Buy
ChemScene CS-5917 Relugolix >98.0% 5mg $120 2021-12-16 Buy
ChemScene CS-5917 Relugolix >98.0% 10mg $190 2021-12-16 Buy
ChemScene CS-5917 Relugolix >98.0% 50mg $660 2021-12-16 Buy
ChemScene CS-5917 Relugolix >98.0% 100mg $1100 2021-12-16 Buy
Crysdot CD11064717 Relugolix(TAK385) 97% 5mg $245 2021-12-16 Buy
Crysdot CD11064717 Relugolix(TAK385) 97% 10mg $350 2021-12-16 Buy

Properties

Melting point :228 °C (decomp)(Solv: ethyl acetate (141-78-6); tetrahydrofuran (109-99-9))
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O

Safety Information

Symbol(GHS): GHS hazard pictograms
Signal word: Warning
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
H361 Suspected of damaging fertility or the unborn child Reproductive toxicity Category 2 Warning P201, P202, P281, P308+P313, P405,P501
H371 May cause damage to organs Specific target organ toxicity, single exposure Category 2 Warning P260, P264, P270, P309+P311, P405,P501
Precautionary statements:
P201 Obtain special instructions before use.
P202 Do not handle until all safety precautions have been read and understood.
P260 Do not breathe dust/fume/gas/mist/vapours/spray.
P264 Wash hands thoroughly after handling.
P264 Wash skin thouroughly after handling.
P270 Do not eat, drink or smoke when using this product.
P281 Use personal protective equipment as required.
P308+P313 IF exposed or concerned: Get medical advice/attention.
P309+P311 IF exposed or if you feel unwell: call a POISON CENTER or doctor/physician.
P405 Store locked up.
P501 Dispose of contents/container to..…

Description

Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. It possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.

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