| Identification | Back Directory | [Name]
PF-3246799 hydrochloride | [CAS]
1065114-52-4 | [Synonyms]
PF-3246799 hydrochloride
PF-03246799 hydrochloride
PF-03246799 hydrochloride >=98% (HPLC)
6,7,8,9-Tetrahydro-2-(phenylmethyl)-5H-pyrimido[4,5-d]azepine hydrochloride | [Molecular Formula]
C15H18ClN3 | [MDL Number]
MFCD28347837 | [MOL File]
1065114-52-4.mol | [Molecular Weight]
275.78 |
| Chemical Properties | Back Directory | [storage temp. ]
room temp | [solubility ]
H2O: soluble20mg/mL, clear | [form ]
powder | [color ]
white to beige | [Water Solubility ]
H2O: 20mg/mL, clear |
| Hazard Information | Back Directory | [Biological Activity]
PF-3246799 is a potent serotonin 5-HT2C receptor agonist with an EC50 of 4.5 nM and minimal activity at 5-HT2A and 5-HT2B receptors. PF-3246799 had good efficacy in a preclinical canine model of stress urinary incontinence. |
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| Company Name: |
Energy Chemical
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| Tel: |
021-58432009 400-005-6266 |
| Website: |
http://www.energy-chemical.com |
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