| Identification | Back Directory | [Name]
BET-IN-1 | [CAS]
1422554-34-4 | [Synonyms]
BET-IN-1
I-BET282
BET inhibitor 1
1H-Imidazo[4,5-c]quinoline, 7-(3,5-dimethyl-4-isoxazolyl)-8-methoxy-1-[(1R)-2-methoxy-1-methylethyl]-2-(tetrahydro-2H-pyran-4-yl)- | [Molecular Formula]
C25H30N4O4 | [MDL Number]
MFCD29924729 | [MOL File]
1422554-34-4.mol | [Molecular Weight]
450.53 |
| Hazard Information | Back Directory | [Description]
BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1, compound example 2, has a plC50 in the range 6.0 - 7.0.IC50 value: 6.0 - 7.0 (plC50)Target: bromodomain | [storage]
Store at -20°C | [References]
[1]. Demont Emmanuel Hubert, et al. Preparation of 4-(8-methoxy-1-(1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole, its salts and isomers and their use as bromodomain inhibitors. From PCT Int. Appl. (201 |
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| Company Name: |
Musechem
|
| Tel: |
+1-800-259-7612 |
| Website: |
www.musechem.com |
| Company Name: |
BOC Sciences
|
| Tel: |
16314854226 |
| Website: |
www.bocsci.com |
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