| Identification | Back Directory | [Name]
AM2201 N-(4-hydroxypentyl) metabolite | [CAS]
1427521-34-3 | [Synonyms]
AM-2201 4-hydroxypenty metabolite
AM-2201 4-hydroxypentyl metabolite
AM2201 N-(4-hydroxypentyl) metabolite
[1-(5-fluoro-4-hydroxypentyl)indol-3-yl]-naphthalen-1-ylmethanone
(1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl)(naphthalen-1-yl)methanone | [Molecular Formula]
C24H22FNO2 | [MDL Number]
MFCD32672185 | [MOL File]
1427521-34-3.mol | [Molecular Weight]
375.44 |
| Hazard Information | Back Directory | [Description]
AM2201 is a potent synthetic cannabinoid (CB) with Ki values of 1.0 and 2.6 nM for the CB1 and CB2 receptors, respectively.1 AM2201 N-(4-hydroxypentyl) metabolite is an expected urinary metabolite of AM2201, based on the known metabolism of similar compounds.2 Its biological actions are unknown. | [Uses]
4-Hydroxypentyl AM-2201 is a metabolite of AM-2201 (A575830), is a drug which acts as a potent but unselective agonist for the cannabinoid receptor CB1 or CB2. | [References]
1. Makriyannis, A., and Deng, H. Cannabimimetic indole derivatives US7241799B2,(2001).
2. Wintermeyer, A., M?ller, I., Thevis, M., et al. In vitro phase I metabolism of the synthetic cannabimimetic JWH-018 Anal. Bioanal. Chem. 398(5),2141-2153(2010). |
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Energy Chemical
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