| Identification | Back Directory | [Name]
PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO- | [CAS]
152811-62-6 | [Synonyms]
CS-2135
Sb207256
SB 207266
PIBOSEROD
Piboserod [inn]
Unii-4uq3S81B25
SB207266(Piboserod)
Piboserod(SB-207266)
SB-207266 >=98% (HPLC)
SB-207266;SB 207266;SB207266
N-[(1-Butyl-4-piperidinyl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a]indole-10-carboxamide
N-[(1-butylpiperidin-4-yl)methyl]-3,4-dihydro-2H-[1,3]oxazino[3,2-a]indole-10-carboxamide
2H-[1,3]Oxazino[3,2-a]indole-10-carboxamide,N-[(1-butyl-4-piperidinyl)methyl]-3,4-dihydro-
PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO- | [Molecular Formula]
C22H31N3O2 | [MDL Number]
MFCD00923681 | [MOL File]
152811-62-6.mol | [Molecular Weight]
369.5 |
| Chemical Properties | Back Directory | [Melting point ]
110-113° | [Boiling point ]
570.3±35.0 °C(Predicted) | [density ]
1.22±0.1 g/cm3(Predicted) | [storage temp. ]
2-8°C | [solubility ]
DMF: 30 mg/mL; DMSO: 20 mg/mL; Ethanol: 30 mg/mL; Ethanol:PBS (pH7.2)(1:20): 0.05 mg/mL | [form ]
powder | [pka]
13.86±0.20(Predicted) | [color ]
white to beige |
| Hazard Information | Back Directory | [Uses]
Treatment
of irritable bowel syndrome (selective 5HT4receptor
antagonist). | [Biochem/physiol Actions]
SB-207266 is a potent, selective, orally active and long-acting 5-HT4 antagonist in vivo. | [storage]
Store at -20°C |
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