Identification | Back Directory | [Name]
T-3764518 | [CAS]
1809151-56-1 | [Synonyms]
T-3764518 1,3,4-Oxadiazole-2-methanol, 5-[6-[4-(trifluoromethyl)-4-[4-(trifluoromethyl)phenyl]-1-piperidinyl]-3-pyridazinyl]- | [Molecular Formula]
C20H17F6N5O2 | [MDL Number]
MFCD31813612 | [MOL File]
1809151-56-1.mol | [Molecular Weight]
473.37 |
Chemical Properties | Back Directory | [storage temp. ]
4°C, away from moisture and light | [solubility ]
DMSO : 95 mg/mL (200.69 mM; Need ultrasonic) | [form ]
Solid | [color ]
White to off-white |
Hazard Information | Back Directory | [Biological Activity]
T-3764518 is a novel and potent stearoyl coenzyme A desaturase (SCD) inhibitor with an IC50 of 4.7 nM. | [References]
[1]. Imamura K, et al. Discovery of Novel and Potent Stearoyl Coenzyme A Desaturase 1 (SCD1) Inhibitors as Anticancer Agents. Bioorg Med Chem. 2017 Jul 15;25(14):3768-3779. |
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