| Identification | Back Directory | [Name]
(S)-2-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-ylcarbamoyl)-4-methylpenty((R)-1-amino-3-phenylpropyl)phosphinic acid | [CAS]
2007955-07-7 | [Synonyms]
(S)-2-((S)-1-AMINO-3-(1H-INDOL-3-YL)-1-OXOPROPAN-2-YLCARBAMOYL)-4-METHYLPENTY((R)-1-AMINO-3-PHENYLPR
(S)-2-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-ylcarbamoyl)-4-methylpenty((R)-1-amino-3-phenylpropyl)phosphinic acid | [Molecular Formula]
C27H37N4O4P | [MOL File]
2007955-07-7.mol | [Molecular Weight]
512.58 |
| Hazard Information | Back Directory | [Description]
DG013A is a a phosphinic pseudotripeptide and ERAP2 inhibitor with nanomolar potency for ERAP2. A crystal structure of a phosphinic pseudotripeptide (DG013A) bound into the active site of ERAP2 revealed five distinct protein elements that were hypothesized to drive inhibitor potency. |
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