Identification | Back Directory | [Name]
BENZOTRIPT | [CAS]
39544-74-6 | [Synonyms]
benzotripte BENZOTRIPT USP/EP/BP Nα-(4-Chlorobenzoyl)-L-tryptophan L-Tryptophan, N-(4-chlorobenzoyl)- (S)-α-(4-Chlorobenzoylamino)-1H-indole-3-propionic acid | [EINECS(EC#)]
254-500-0 | [Molecular Formula]
C18H15ClN2O3 | [MOL File]
39544-74-6.mol | [Molecular Weight]
342.78 |
Chemical Properties | Back Directory | [storage temp. ]
-20°C | [solubility ]
Soluble in DMSO (up to at least 25 mg/ml) | [form ]
solid | [color ]
White | [Stability:]
Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months. |
Hazard Information | Back Directory | [Description]
Benzotript (39544-74-6) antagonizes the interaction of cholecystokinin and related peptides with the cholecystokinin receptor.1 ?It has been reported to potentiate morphine analgesia via interaction with opioid receptors.2 | [Uses]
Benzotript is an antiulcer drug that is a cholecystokinin receptor (CCK-2R) antagonist . | [References]
1) Hahne (1981), Proglumide and benzotript: Members of a different class of cholecystokinin receptor antagonists; Proc. Natl. Acad. Sci. USA. 78 6304
2) Gaudreau et al. (1990), Cholecystokinin antagonists proglumide, lorglumide and benzotript, but not L-364,718, interact with brain opioid binding sites; Neuropeptides 16 51 |
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Company Name: |
Enamine
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Tel: |
(380) 44 537 32 18 |
Website: |
www.enamine.net |
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