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2171388-28-4

英文名称 Spiro[3H-indole-3,4'-piperidin]-2(1H)-one, 6-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-4-fluoro-1'-(3,4,5,6,7,8-hexahydro-8-methyl-4-oxopyrido[2,3-d]pyrimidin-2-yl)-1-methyl-, rel-
CAS 2171388-28-4
分子式 C27H35FN6O3
分子量 510.6
MOL 文件 2171388-28-4.mol
2171388-28-4 结构式 2171388-28-4 结构式

基本信息

英文别名
Spiro[3H-indole-3,4'-piperidin]-2(1H)-one, 6-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-4-fluoro-1'-(3,4,5,6,7,8-hexahydro-8-methyl-4-oxopyrido[2,3-d]pyrimidin-2-yl)-1-methyl-, rel-

应用领域

用途一
RK-582 is an orally efficacious spiroindolinone-based tankyrase inhibitor for the treatment of colon cancer. It exhibits a markedly improved robust tumor growth inhibition in a COLO-320DM mouse xenograft model when orally administered.
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