2750001-23-9
中文名称
AZD0095
英文名称
INDEX NAME NOT YET ASSIGNED
CAS
2750001-23-9
分子式
C27H32N8O2
分子量
500.61
MOL 文件
2750001-23-9.mol
更新日期
2023/08/17 14:26:57
2750001-23-9 结构式
应用领域
用途一
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology. AZD0095 has excellent potency (1.3 nM), MCT1 selectivity (>1000×), secondary pharmacology, clean mechanism of action, suitable properties for oral administration in the clinic, and good preclinical efficacy in combination with cediranib.