苯赖加压素乙酸酯
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- CAS号:
- 914453-97-7
- 英文名:
- Felypressin Acetate
- 英文别名:
- Oxytocin Impurity 12
- 中文名:
- 苯赖加压素乙酸酯
- 中文别名:
- 苯赖加压素乙酸酯;苯赖加压素乙酸盐;催产素杂质 12;N-[5-氨基-1-(氨基甲酰基甲基氨基甲酰基)戊基]-1-[19-氨基-13,16-二苄基-10-(2-氨基甲酰基乙基)-7-(氨基甲酰基甲基)-6,9,12,15,18-五氧代-1,2-二硫-5,8,11,14,17-五氮杂环二十烷-4-羰基]吡咯烷-2-羧酰胺乙酸盐
- CBNumber:
- CB02695879
- 分子式:
- C48H69N13O13S2
- 分子量:
- 1100.28
- MOL File:
- 914453-97-7.mol
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苯赖加压素乙酸酯化学性质
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储存条件:
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Store at -20°C
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形态:
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Solid
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颜色:
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White to off-white
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水溶解性:
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Water : 100 mg/mL (Need ultrasonic)
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苯赖加压素乙酸酯性质、用途与生产工艺
Felypressin acetate (PLV-2 acetate) 是一种非儿茶酚胺的血管收缩剂，也是一种加压素 1 (vasopressin 1) 激动剂。Felypressin acetate 广泛用于牙科手术中。
Felypressin is a synthetic hormone of the posterior pituitary lobe characterized by vasoconstrictor properties that is widely used in dental procedures. The vasoconstrictor action of Felypressin seems to be mediated by V1 receptors of the blood vessel smooth muscle cells.
Felypressin can reduce toxicity during dental procedures. Felypressin increases the diastolic blood pressure of hypertensive patients with controlled blood pressure.
Cardiovascular effects of Felypressin (240 ng/kg; intravenous injection) are studied in Wistar rats. Felypressin induces a pressor effect. Felypressin depends on V1 receptors to induce pressor and bradycardic effects, and that it produces a high relationship between bradycardia and mean arterial pressure variation depending on area postrema and central V1 receptors.
苯赖加压素乙酸酯
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914453-97-7, 苯赖加压素乙酸酯 相关搜索:
- Amino Acids & Derivatives, Pharmaceuticals, Intermediates & Fine Chemicals
- 抑制剂
- 药靶配体
- 苯赖加压素乙酸盐
- 催产素杂质 12
- N-[5-氨基-1-(氨基甲酰基甲基氨基甲酰基)戊基]-1-[19-氨基-13,16-二苄基-10-(2-氨基甲酰基乙基)-7-(氨基甲酰基甲基)-6,9,12,15,18-五氧代-1,2-二硫-5,8,11,14,17-五氮杂环二十烷-4-羰基]吡咯烷-2-羧酰胺乙酸盐
- 苯赖加压素乙酸酯
- 914453-97-7
- Oxytocin Impurity 12