BB-Cl-Amidine hydrochloride
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- CAS号:
- 英文名:
- BB-Cl-Amidine hydrochloride
- 英文别名:
- BB-Cl-Amidine hydrochloride
- 中文名:
- BB-Cl-Amidine hydrochloride
- 中文别名:
- 化合物 T10482L
- CBNumber:
- CB05419683
- 分子式:
- C??H??Cl?N?O
- 分子量:
- 0
- MOL File:
- Mol file
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BB-Cl-Amidine hydrochloride化学性质
BB-Cl-Amidine hydrochloride性质、用途与生产工艺
BB-Cl-Amidine hydrochloride 是肽基精氨酸脱胺酶 (PAD) 的抑制剂。
Treatment with BB-Cl-amidine subtly reduces splenomegaly in MRL/lpr mice, while there is a trend towards increased circulating levels of anti-NET antibodies with PAD inhibitor treatment. However, neither PAD inhibitor affected body weight or total IgG levels. Indeed, treatment with both Cl-amidine and BB-Cl-amidine significantly improves endothelium-dependent vasorelaxation. The BB-Cl-amidine group also shows a strong trend towards downregulation of IRGs. Treatment with either Cl-amidine or BB-Cl-amidine significantly improves muzzle alopecia, in many cases preventing it entirely.
Animal Model:
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MRL/lpr mice.
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Dosage:
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1 mg/kg.
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Administration:
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Subcutaneous injection daily from 8 to 14 weeks of age.
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Result:
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Significantly improved endothelium-dependent vasorelaxation and showed a strong trend towards downregulation of IRGs.
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BB-Cl-Amidine hydrochloride
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上游原料
下游产品
BB-Cl-Amidine hydrochloride 试剂级价格
更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
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2024/08/19 | HY-111347A | BB-Cl-Amidine hydrochloride BB-Cl-Amidine hydrochloride | | 1mg | 450元 |
2024/08/19 | HY-111347A | BB-Cl-Amidine hydrochloride BB-Cl-Amidine hydrochloride | | 5mg | 950元 |
BB-Cl-Amidine hydrochloride
生产厂家
BB-Cl-Amidine hydrochloride 相关搜索:
- 化合物 T10482L
- BB-Cl-Amidine hydrochloride