7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
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- CAS号:
- 179248-59-0
- 英文名:
- 6,7-Dimethoxy-N-(4-phenoxyphenyl)-
- 英文别名:
- Edr;HHAT;HB-1;Mar2;MART2;SKI-1;MEF3L;Src I1;Src-l1;Src Inhibitor-1
- 中文名:
- 7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
- 中文别名:
- SRC抑制剂1;化合物SRC INHIBITOR 1;7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉;6,7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉;6,7-二甲氧基-N-(4-苯氧基苯基)喹唑啉-4-胺;6,7-二甲氧基-N-(4-苯氧基苯基)-4-喹唑啉胺;双位点SRC酪氨酸激酶抑制剂(SRC INHIBITOR 1)
- CBNumber:
- CB22508388
- 分子式:
- C22H19N3O3
- 分子量:
- 373.4
- MOL File:
- 179248-59-0.mol
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7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉化学性质
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储存条件:
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2-8°C
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溶解度:
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DMSO: >10mg/mL
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形态:
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white powder
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颜色:
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White or off-white
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稳定性:
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Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 week.
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7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉性质、用途与生产工艺
Src Inhibitor 1是Src和Lck的竞争性抑制剂，IC50分别为44 nM和88 nM。它也能抑制Csk和Yes。
| Target | Value |
Src
(Cell-free assay)
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44 nM
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Lck
(Cell-free assay)
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88 nM
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Src-I1 is competitive with both ATP and peptide binding sites of the kinase. The IC
50
values are 44 and 88 nM for Src and Lck, respectively. Src-I1, is found to be a potent inhibitor of Src (IC
50
=0.18 μM), but also inhibited other Src family members, such as Lck, Csk and Yes with similar potency to Src, and RIP2 (IC
50
=0.026 μM) with even greater potency. In addition, it inhibited CHK2 with similar potency to Src, and Aurora B with slightly lower potency.
7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
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| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/11/08 | HY-101053 | 7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
Src Inhibitor 1 | 179248-59-0 | 2mg | 500元 |
| 2024/11/08 | HY-101053 | 7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
Src Inhibitor 1 | 179248-59-0 | 10mM * 1mLin DMSO | 575元 |
7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
生产厂家
179248-59-0, 7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉 相关搜索:
- Inhibitors
- Heterocycles
- Aromatics
- Amines
- 抑制剂
- 合成有机化合物配体
- 标准品
- 细胞生物学试剂
- 合成
- 6,7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
- 6,7-二甲氧基-N-(4-苯氧基苯基)喹唑啉-4-胺
- 化合物SRC INHIBITOR 1
- SRC抑制剂1
- 6,7-二甲氧基-N-(4-苯氧基苯基)-4-喹唑啉胺
- 双位点SRC酪氨酸激酶抑制剂(SRC INHIBITOR 1)
- 7-二甲氧基-N-(4-苯氧基苯基)- 氨基喹唑啉
- 179248-59-0
- Src-I1
Src Inhibitor 1
- Src Inhibitor 1,Src Kinase Inhibitor1,Src,Inhibitor,Src Kinase Inhibitor-1,Src Inhibitor1,inhibit,Src Inhibitor-1
- 6,7-Dimethoxy-N-(4-phenoxyphenyl)-aminoquinazoline
- 4-Quinazolinamine, 6,7-dimethoxy-N-(4-phenoxyphenyl)-
- Src Kinase Inhibitor 1
- 46,7-Dimethoxy-N-(4-phenoxyphenyl)-
- Src Kinase Inhibitor I - CAS 179248-59-0 - Calbiochem
- 6,7-dimethoxy-N-(4-phenoxyphenyl)quinazolin-4-amine
- Monoclonal Anti-PEG10 antibody produced in mouse
- MEF3L
- Mar2
- HB-1
- Edr
- Protein-cysteine N-palmitoyltransferase HHAT
- MART2
- HHAT
- ANTI-HHAT (N-TERM) antibody produced in rabbit
- Src-l1
- Src Inhibitor-1
- SKI-1
- Src I1
- 6,7-Dimethoxy-N-(4-phenoxyphenyl)-