fluphenazine O-enantate
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- CAS号:
- 2746-81-8
- 英文名:
- fluphenazine O-enantate
- 英文别名:
- moditen enanthate;fluphenazine O-enantate;Fluphenazine enantate CRS;Fluphenazine Decanoate Impurity 3 (Fluphenazine Decanoate EP Impurity C);2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]propyl]piperazin-1-yl]ethyl heptanoate;2-[4-[3-[2-(Trifluoromethyl)phenothiazin-10-yl]propyl]-1-piperazinyl]ethyl heptanoate;enanthic acid 2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]propyl]piperazin-1-yl]ethyl ester;Heptanoic acid, 2-4-3-2-(trifluoromethyl)-10H-phenothiazin-10-ylpropyl-1-piperazinylethyl ester
- 中文名:
- fluphenazine O-enantate
- 中文别名:
- 氟奋乃静酯;氟奋乃静庚酸酯;化合物 T11304;癸氟奋乃静杂质C(EP);氟奋乃静庚酸盐 EP标准品;氟奋乃静癸酸酯杂质C (EP);癸氟奋乃静杂质3(癸氟奋乃静EP杂质C);2-[4-[3-[2-(三氟甲基)吩噻嗪-10-基]丙基]哌嗪-1-基]乙基庚酸酯
- CBNumber:
- CB2935054
- 分子式:
- C29H38F3N3O2S
- 分子量:
- 549.698
- MOL File:
- 2746-81-8.mol
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fluphenazine O-enantate化学性质
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熔点:
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184.5°C
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沸点:
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629.4±55.0 °C(Predicted)
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密度:
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1.1661 (estimate)
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溶解度:
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Practically insoluble in water, very soluble in ethanol and in methylene chloride, freely soluble in methanol.
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酸度系数(pKa):
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7.32±0.10(Predicted)
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fluphenazine O-enantate性质、用途与生产工艺
Fluphenazine enanthate 是第一种长效抗精神病药物，用于研究精神分裂症。
Fluphenazine enanthate (2,4, 8 mg/kg; IM) significant inhibition of the avoidance performance is observed as long as 16, 23, and 28 days, respectively.
Fluphenazine enanthate (8 mg/kg) drinking behavior is almost completely suppressed for 24 hours immediately following the administration.
Fluphenazine enanthate (8 mg/kg) produces transient body weight Iosses in the rats.
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Animal Model:
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Fifty-four male adult rats of Wistar strain
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Dosage:
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2, 4, and 8 mg/kg
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Administration:
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Index medicus (IM )
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Result:
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Three doses of Fluphenazine enanthate significant inhibition of the avoidance performance was observed as long as 16, 23, and 28 days, respectively.
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fluphenazine O-enantate
上下游产品信息
上游原料
下游产品
fluphenazine O-enantate
生产厂家
2746-81-8, fluphenazine O-enantate 相关搜索:
- Organics
- 氟奋乃静酯
- 化合物 T11304
- 2-[4-[3-[2-(三氟甲基)吩噻嗪-10-基]丙基]哌嗪-1-基]乙基庚酸酯
- 癸氟奋乃静杂质3(癸氟奋乃静EP杂质C)
- 氟奋乃静庚酸盐 EP标准品
- 癸氟奋乃静杂质C(EP)
- 氟奋乃静癸酸酯杂质C (EP)
- 氟奋乃静庚酸酯
- 2746-81-8
- Fluphenazine Decanoate Impurity 3 (Fluphenazine Decanoate EP Impurity C)
- Fluphenazine enantate CRS
- 2-[4-[3-[2-(Trifluoromethyl)phenothiazin-10-yl]propyl]-1-piperazinyl]ethyl heptanoate
- enanthic acid 2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]propyl]piperazin-1-yl]ethyl ester
- 2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]propyl]piperazin-1-yl]ethyl heptanoate
- moditen enanthate
- Heptanoic acid, 2-4-3-2-(trifluoromethyl)-10H-phenothiazin-10-ylpropyl-1-piperazinylethyl ester
- fluphenazine O-enantate