TLX agonist 1
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- CAS号:
- 958323-31-4
- 英文名:
- TLX agonist 1
- 英文别名:
- CCRP2;TLX agonist 1;TLX a onist 1;(4-Benzhydrylpiperazin-1-yl)(1,5-dimethyl-1H-pyrazol-3-yl)methanone;Methanone, (1,5-dimethyl-1H-pyrazol-3-yl)[4-(diphenylmethyl)-1-piperazinyl]-;TLX agonist-1,transcriptional,TLX agonist 1,repressive,Inhibitor,ligand,inhibit,TLX agonist1,orphan
- 中文名:
- TLX agonist 1
- 中文别名:
- TLX激动剂1;化合物TLX AGONIST 1;(4-苯甲酰基哌嗪-1-基)(1,5-二甲基-1H-吡唑-3-基)甲酮
- CBNumber:
- CB35832809
- 分子式:
- C23H26N4O
- 分子量:
- 374.48
- MOL File:
- 958323-31-4.mol
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TLX agonist 1化学性质
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沸点:
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539.6±50.0 °C(Predicted)
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密度:
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1.16±0.1 g/cm3(Predicted)
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储存条件:
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2-8°C
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溶解度:
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DMSO: 62.5 mg/mL (166.90 mM)
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酸度系数(pKa):
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5.78±0.10(Predicted)
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形态:
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Solid
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颜色:
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White to off-white
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TLX agonist 1性质、用途与生产工艺
TLX agonist 1 (CCRP2, SUN23314) 是一种 orphan nuclear receptor tailless (TLX, NR2E1) 的调节剂，其EC50值为1.0 μM，Kd值为650 nM。TLX agonist 1 (CCRP2, SUN23314) 与重组TLX蛋白结合并增强TLX转录抑制活性。
| Target | Value |
NR2E1
(Cell-free assay)
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650 nM(Kd)
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NR2E1
(Cell-free assay)
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1.0 μM(EC50)
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TLX agonist 1
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/11/08 | HY-135572 | TLX agonist 1
TLX agonist 1 | 958323-31-4 | 1mg | 500元 |
| 2024/11/08 | HY-135572 | TLX agonist 1
TLX agonist 1 | 958323-31-4 | 5mg | 1100元 |
958323-31-4, TLX agonist 1 相关搜索:
- 药靶配体
- 抑制剂
- TLX激动剂1
- 化合物TLX AGONIST 1
- (4-苯甲酰基哌嗪-1-基)(1,5-二甲基-1H-吡唑-3-基)甲酮
- 958323-31-4
- TLX a onist 1
- TLX agonist-1,transcriptional,TLX agonist 1,repressive,Inhibitor,ligand,inhibit,TLX agonist1,orphan
- CCRP2
- (4-Benzhydrylpiperazin-1-yl)(1,5-dimethyl-1H-pyrazol-3-yl)methanone
- Methanone, (1,5-dimethyl-1H-pyrazol-3-yl)[4-(diphenylmethyl)-1-piperazinyl]-
- TLX agonist 1