CCK-B RECEPTOR ANTAGONIST 2
|
|
|
- CAS号:
- 155412-88-7
- 英文名:
- CCK-B Receptor Antagonist 2
- 英文别名:
- CCK-B Receptor Antagonist 2;CCK B Receptor Antagonist 2,CCKB Receptor Antagonist 2;Urea, N-(3-aminophenyl)-N'-[(3R)-1-(3,3-dimethyl-2-oxobutyl)-2,3-dihydro-2-oxo-5-(2-pyridinyl)-1H-1,4-benzodiazepin-3-yl]-
- 中文名:
- CCK-B RECEPTOR ANTAGONIST 2
- 中文别名:
- 化合物 T10707
- CBNumber:
- CB65821330
- 分子式:
- C27H28N6O3
- 分子量:
- 484.55
- MOL File:
- 155412-88-7.mol
|
|
|
CCK-B RECEPTOR ANTAGONIST 2化学性质
-
沸点:
-
725.1±60.0 °C(Predicted)
-
|
-
密度:
-
1.29±0.1 g/cm3(Predicted)
-
|
-
储存条件:
-
Store at -20°C
-
|
-
溶解度:
-
DMSO: 250 mg/mL (515.94 mM)
-
|
-
酸度系数(pKa):
-
11.35±0.40(Predicted)
-
|
-
形态:
-
Solid
-
|
-
颜色:
-
White to light yellow
-
|
CCK-B RECEPTOR ANTAGONIST 2性质、用途与生产工艺
CCK-B Receptor Antagonist 2，化合物 15b，是有效的口服活性 Gastrin/CCK-B 拮抗剂，IC50 值为 0.43 nM。 CCK-B Receptor Antagonist 2 还抑制 Gastrin/CCK-A 活性，IC50 为 1.82 μM。
IC50: 0.43 nM (Gastrin/CCK-B); 1.82 μM (Gastrin/CCK-A)
CCK-B Receptor Antagonist 2 (0.1 μmol/kg; intravenous injection) has an inhibition effect on pentagastrin-induced gastric acid secretion in anethsetized rats with an ED
50
of 8.3 nmol/kg.
CCK-B RECEPTOR ANTAGONIST 2
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/04/30 | HY-129357 | CCK-B Receptor Antagonist 2 | | 1 mg | 2045元 |
| 2024/04/30 | HY-129357 | CCK-B RECEPTOR ANTAGONIST 2
CCK-B Receptor Antagonist 2 | 155412-88-7 | 5mg | 4500元 |
CCK-B RECEPTOR ANTAGONIST 2
生产厂家
155412-88-7, CCK-B RECEPTOR ANTAGONIST 2 相关搜索:
- 化合物 T10707
- 155412-88-7
- Urea, N-(3-aminophenyl)-N'-[(3R)-1-(3,3-dimethyl-2-oxobutyl)-2,3-dihydro-2-oxo-5-(2-pyridinyl)-1H-1,4-benzodiazepin-3-yl]-
- CCK B Receptor Antagonist 2,CCKB Receptor Antagonist 2
- CCK-B Receptor Antagonist 2