H4 RECEPTOR ANTAGONIST 1
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- CAS号:
- 848217-00-5
- 英文名:
- 8-chloro-2-methyl-4-(4-methylpiperazin-1-yl)-[1]benzofuro[3,2-d]pyrimidine
- 英文别名:
- H4 Receptor antagonist 1;Benzofuro[3,2-d]pyrimidine, 8-chloro-2-methyl-4-(4-methyl-1-piperazinyl)-;8-chloro-2-methyl-4-(4-methylpiperazin-1-yl)-[1]benzofuro[3,2-d]pyrimidine;inhibit,Inhibitor,Histamine Receptor,H4 Receptor antagonist 1,H-4 Receptor antagonist 1
- 中文名:
- H4 RECEPTOR ANTAGONIST 1
- 中文别名:
- 化合物H4 RECEPTOR ANTAGONIST 1
- CBNumber:
- CB74603190
- 分子式:
- C16H17ClN4O
- 分子量:
- 316.79
- MOL File:
- 848217-00-5.mol
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H4 RECEPTOR ANTAGONIST 1化学性质
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密度:
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1.328±0.06 g/cm3(Predicted)
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储存条件:
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Store at -20°C
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溶解度:
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DMSO : 10 mg/mL (31.57 mM)
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形态:
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Solid
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酸度系数(pKa):
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6.73±0.42(Predicted)
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颜色:
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White to off-white
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H4 RECEPTOR ANTAGONIST 1性质、用途与生产工艺
H4 Receptor antagonist 1 是一种有效的、有选择性的组胺H4受体 (H4R) 的反向激动剂，其IC50 值为19 nM。
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H
4
receptor
19 nM (IC
50
)
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H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC
50
of 19 nM.
H4 Receptor antagonist 1 indicates that metabolic stability in rat microsomes is very low with only 1% parent compound remaining after 10 min incubation.
H4 RECEPTOR ANTAGONIST 1
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/04/30 | HY-114025 | H4 RECEPTOR ANTAGONIST 1
H4 Receptor antagonist 1 | 848217-00-5 | 5mg | 750元 |
| 2024/04/30 | HY-114025 | H4 RECEPTOR ANTAGONIST 1
H4 Receptor antagonist 1 | 848217-00-5 | 10mM * 1mLin DMSO | 825元 |
H4 RECEPTOR ANTAGONIST 1
生产厂家
848217-00-5, H4 RECEPTOR ANTAGONIST 1 相关搜索:
- 化合物H4 RECEPTOR ANTAGONIST 1
- 848217-00-5
- inhibit,Inhibitor,Histamine Receptor,H4 Receptor antagonist 1,H-4 Receptor antagonist 1
- Benzofuro[3,2-d]pyrimidine, 8-chloro-2-methyl-4-(4-methyl-1-piperazinyl)-
- H4 Receptor antagonist 1
- 8-chloro-2-methyl-4-(4-methylpiperazin-1-yl)-[1]benzofuro[3,2-d]pyrimidine