PDK1 INHIBITOR
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- CAS号:
- 850717-64-5
- 英文名:
- PDK1 Inhibitor
- 英文别名:
- BX-517;BIX517;CS-1693;BX-517;BX 517;PDK1 Inhibitor 2;PDK1 Inhibitor II;BX517, 10 mM in DMSO;BX517(PDK1 inhibitor2);inhibit,BX517,Inhibitor,PDK-1;5-Ureido-3-[1-(pyrrol-2-yl)ethylidene]indolin-2-one
- 中文名:
- PDK1 INHIBITOR
- 中文别名:
- 化合物BX517;PDK1抑制剂(BX517);化合物BX517,10 MM DMSO 溶液;5-脲基-3-[1-(吡咯-2-基)亚乙基]吲哚啉-2-酮
- CBNumber:
- CB92667655
- 分子式:
- C15H14N4O2
- 分子量:
- 282.3
- MOL File:
- 850717-64-5.mol
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PDK1 INHIBITOR化学性质
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储存条件:
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Store at -20°C
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溶解度:
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insoluble in H2O; insoluble in EtOH; ≥8.55 mg/mL in DMSO
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形态:
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solid
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颜色:
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Light yellow to khaki
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PDK1 INHIBITOR性质、用途与生产工艺
BX517 是一种有效的，选择性的 PDK1 抑制剂，IC50 值为 6 nM。
BX-517 blocks activation of Akt in tumor cells, is potent with IC
50
of 0.1-1.0 μM. BX-517 blocks AKT2 activation in cells with submicromolar potency. BX-517 is 100-fold selective or better against a panel of seven additional Ser/Thr and Tyr kinases.
PDK1 INHIBITOR
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
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| 2024/11/08 | HY-13842 | BX517 | | 1 mg | 300元 |
| 2024/11/08 | HY-13842 | PDK1 INHIBITOR
BX517 | 850717-64-5 | 5mg | 750元 |
850717-64-5, PDK1 INHIBITOR 相关搜索:
- 抑制剂
- 对照品
- 细胞生物学试剂
- 化合物BX517,10 MM DMSO 溶液
- 化合物BX517
- PDK1抑制剂(BX517)
- 5-脲基-3-[1-(吡咯-2-基)亚乙基]吲哚啉-2-酮
- 850717-64-5
- BX517, 10 mM in DMSO
- {2-oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]-2,3-dihydro-1H-indol-5-yl}urea
- BIX517
- inhibit,BX517,Inhibitor,PDK-1
- 2-Oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]indolin-5-yl]urea,BX-517
- Urea, N-[2,3-dihydro-2-oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]-1H-indol-5-yl]-
- Urea, [2,3-dihydro-2-oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]-1H-indol-5-yl]-
- BX-517;BX 517
- PDK1 Inhibitor II
- CS-1693
- PDK1 Inhibitor 2
- 5-Ureido-3-[1-(pyrrol-2-yl)ethylidene]indolin-2-one
- BX517(PDK1 inhibitor2)
- BX-517