863115-70-2
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- CAS号:
- 863115-70-2
- 英文名:
- MCHr1 antagonist 2
- 英文别名:
- MCHr1 antagonist 2;4H-1-Benzopyran-2-carboxamide, N-[1-(1,3-benzodioxol-5-ylmethyl)-4-piperidinyl]-6-fluoro-4-oxo-;inhibit,Potassium Channel,MCHR1 antagonist 2,IMR-32,melanin,hormone,Melanin concentrating hormone receptor 1,MCHR-1 antagonist 2,hERG,concentrating,MCHR1 (GPR24),Inhibitor,KcsA
- 中文名:
- 863115-70-2
- 中文别名:
- 化合物 T11966;化合物MCHR1 ANTAGONIST 2
- CBNumber:
- CB93384779
- 分子式:
- C23H21FN2O5
- 分子量:
- 424.42
- MOL File:
- 863115-70-2.mol
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863115-70-2化学性质
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储存条件:
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Store at -20°C
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溶解度:
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Soluble in DMSO
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形态:
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Solid
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颜色:
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White to off-white
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863115-70-2性质、用途与生产工艺
MCHR1 antagonist 2 是一种黑色素聚集激素受体 1 (melanin concentrating hormone receptor 1) 拮抗剂，IC50 值为 65 nM；MCHR1 antagonist 2 同时抑制 hERG，在 IMR-32 细胞中，IC50 值为 4.0 nM。
IC50: 65 nM (melanin concentrating hormone receptor 1), 4.0 nM (hERG in IMR-32 cells)
MCHR1 antagonist 2 (Compound 30) is an antagonist of melanin concentrating hormone receptor 1, with an IC
50
of 65 nM. MCHR1 antagonist 2 has inhibitory effects on Ca
2+
flux, and hERG, with IC
50
s of 196 ± 30 nM and 4.0 ± 0.8 nM, respectively, in IMR-32 cells.
863115-70-2
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上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
|---|
| 2024/08/19 | HY-100321 | 863115-70-2
MCHR1 antagonist 2 | 863115-70-2 | 5mg | 1300元 |
| 2024/08/19 | HY-100321 | 863115-70-2
MCHR1 antagonist 2 | 863115-70-2 | 10mg | 2200元 |
863115-70-2, 863115-70-2 相关搜索:
- 化合物MCHR1 ANTAGONIST 2
- 化合物 T11966
- 863115-70-2
- inhibit,Potassium Channel,MCHR1 antagonist 2,IMR-32,melanin,hormone,Melanin concentrating hormone receptor 1,MCHR-1 antagonist 2,hERG,concentrating,MCHR1 (GPR24),Inhibitor,KcsA
- 4H-1-Benzopyran-2-carboxamide, N-[1-(1,3-benzodioxol-5-ylmethyl)-4-piperidinyl]-6-fluoro-4-oxo-
- MCHr1 antagonist 2