PROTAC IRAK4 degrader-8
- CAS No.
- 2911615-06-8
- Chemical Name:
- PROTAC IRAK4 degrader-8
- Synonyms
- PROTAC IRAK4 degrader-8
- CBNumber:
- CB014286601
- Molecular Formula:
- Molecular Weight:
- 0
- MDL Number:
- MOL File:
- Mol file
PROTAC IRAK4 degrader-8 Chemical Properties,Uses,Production
Uses
PROTAC IRAK4 degrader-8 (Compound 2) is a PROTAC IRAK4 degrader (IC50: 15.5 nM). PROTAC IRAK4 degrader-8 degrades IRAK4 in THP-1 cells (DC50: 1.8 nM)。PROTAC IRAK4 degrader-8 also inhibits L-6 production in human whole blood and LPS-induced human PBMC cells, with IC50s of 246 nM and 2.2 nM respectively[1].
References
[1] Ye Zhengqing. IRAK4 degradation agent, preparation method and application thereof. Patent. CN115710274.
[2] Ye Z, et al. Preparation of (pyrazolyl)pyrazolo[1,5-a]pyrimidinyl carboxamide derivatives as IRAK4 degrading agents and its applications. China, CN115710274 A. 2023-02-24.
PROTAC IRAK4 degrader-8 Preparation Products And Raw materials
Raw materials
Preparation Products
PROTAC IRAK4 degrader-8 Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
TargetMol Chemicals Inc. | +8613564774135 | zijue.cai@tsbiochem.com | United States | 19881 | 58 |
TargetMol Chemicals Inc. | 15002134094 | marketing@targetmol.cn | China | 19699 | 58 |
Supplier | Advantage |
---|---|
TargetMol Chemicals Inc. | 58 |
TargetMol Chemicals Inc. | 58 |
View Lastest Price from PROTAC IRAK4 degrader-8 manufacturers
Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
---|---|---|---|---|---|---|---|---|
![]() |
2024-11-19 | PROTAC IRAK4 degrader-8
2911615-06-8
|
US $0.00-0.00 / mg | 10g | TargetMol Chemicals Inc. |
-
- PROTAC IRAK4 degrader-8
2911615-06-8
- US $0.00-0.00 / mg
- TargetMol Chemicals Inc.