ChemicalBook >> CAS DataBase List >>BRD-IN-3
BRD-IN-3
- CAS No.
- 2351938-32-2
- Chemical Name:
- BRD-IN-3
- Synonyms
- BRD-IN-3;BRD IN 3,BRDIN3;4H-Pyrrolo[3,2-d]pyrimidin-4-one, 2-[[(3R,5R)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-3-piperidinyl]amino]-3,5-dihydro-3-methyl-
- CBNumber:
- CB25821291
- Molecular Formula:
- C21H25N5O3
- Molecular Weight:
- 395.45
- MDL Number:
- MFCD32067976
- MOL File:
- 2351938-32-2.mol
Last updated:2023-05-21 10:59:17
BRD-IN-3 Chemical Properties,Uses,Production
Description
BRD-IN-3 ((R,R)-36n) is a highly potent PCAF bromodomain (BRD) inhibitor, with an IC50 of 7 nM. BRD-IN-3 also exhibits activity against GCN5 and FALZ[1]. IC50: PCAF BRD[1].
References
[1]. Huang L, et al. Discovery of Pyrrolo[3,2- d]pyrimidin-4-one Derivatives as a New Class of Potent and Cell-Active Inhibitors of P300/CBP-Associated Factor Bromodomain. J Med Chem. 2019 May 9;62(9):4526-4542.
BRD-IN-3 Preparation Products And Raw materials
Raw materials
Preparation Products
BRD-IN-3 Suppliers
Global( 3)Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | marketing@targetmol.com | United States | 19892 | 58 |
Fan De(Beijing) Biotechnology Co., Ltd. | 15911056312 | liming@bio-fount.com | China | 9730 | 58 |
TargetMol Chemicals Inc. | 15002134094 | marketing@targetmol.cn | China | 19698 | 58 |
Supplier | Advantage |
---|---|
TargetMol Chemicals Inc. | 58 |
Fan De(Beijing) Biotechnology Co., Ltd. | 58 |
TargetMol Chemicals Inc. | 58 |
BRD-IN-3
4H-Pyrrolo[3,2-d]pyrimidin-4-one, 2-[[(3R,5R)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-3-piperidinyl]amino]-3,5-dihydro-3-methyl-
BRD IN 3,BRDIN3
2351938-32-2