Tebipenem
- CAS No.
- 161715-21-5
- Chemical Name:
- Tebipenem
- Synonyms
- LJC11036;LJC-11036;Tebipenem;LJC 11036;Tibipronam;Tebipenem USP/EP/BP;Tebipenem Impurity 5;Tibipenem intermediate 2;inhibit,LJC11036,Bacterial,LJC-11036,Antibiotic,Inhibitor;(4R,5S,6S)-3-[[1-(4,5-Dihydro-2-thiazolyl)-3-azetidinyl]thio]-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
- CBNumber:
- CB52534496
- Molecular Formula:
- C16H21N3O4S2
- Molecular Weight:
- 383.49
- MDL Number:
- MFCD00936545
- MOL File:
- 161715-21-5.mol
- MSDS File:
- SDS
Boiling point | 624.5±65.0 °C(Predicted) |
---|---|
Density | 1.75 |
storage temp. | Sealed in dry,Store in freezer, under -20°C |
solubility | insoluble in EtOH; ≥19.15 mg/mL in H2O with gentle warming; ≥24.9 mg/mL in DMSO |
form | solid |
pka | 4.29±0.60(Predicted) |
color | White to khaki |
FDA UNII | Q2TWQ1I31U |
SAFETY
Risk and Safety Statements
Symbol(GHS) | ![]() GHS07 |
---|---|
Signal word | Warning |
Hazard statements | H302-H315-H319-H335 |
Precautionary statements | P261-P305+P351+P338 |
Tebipenem price
Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|---|
Sigma-Aldrich | SML3203 | Tebipenem ≥98% (HPLC) | 161715-21-5 | 10MG | $81 | 2024-03-01 | Buy |
Sigma-Aldrich | SML3203 | Tebipenem ≥98% (HPLC) | 161715-21-5 | 50MG | $261 | 2024-03-01 | Buy |
ChemScene | CS-3444 | Tebipenem >98.0% | 161715-21-5 | 10mg | $336 | 2021-12-16 | Buy |
ApexBio Technology | B4864 | Tebipenem | 161715-21-5 | 50mg | $594 | 2021-12-16 | Buy |
ChemScene | CS-3444 | Tebipenem >98.0% | 161715-21-5 | 50mg | $900 | 2021-12-16 | Buy |
Tebipenem Chemical Properties,Uses,Production
Biological Activity
tebipenem is an orally available carbapenem antibiotic. tebipenem is active against a panel of clinical isolates from a variety of bacterial species (mic50s ≤ 0.0039 ~ 8 μg/ml), including methicillin-resistant strains of staphylococcus aureus (s. aureus) and staphylococcus epidermidis (s. epidermidis), as well as penicillin-resistant streptococcus pneumoniae (s. pneumonia). tebipenem also inhibits β-lactamase in a time- and concentration-dependent manner. tebipenem pivoxil, a derivative of tebipenem, has been under development as the first orally available carbapenem antibiotic for the treatment of respiratory and otolaryngological infections caused by drug-resistant s. pneumonia in pediatric patients.1. hazra s, xu h, blanchard js. tebipenem, a new carbapenem antibiotic, is a slow substrate that inhibits the β-lactamase from mycobacterium tuberculosis. biochemistry, 2014, 53(22): 3671-3678.2. fujimoto k, takemoto k, hatano k, et al. novel carbapenem antibiotics for parenteral and oral applications: in vitro and in vivo activities of 2-aryl carbapenems and their pharmacokinetics in laboratory animals. antimicrobial agents and chemotherapy, 2013, 57(2): 697-707.
![161715-20-4](/CAS/GIF/161715-20-4.gif)
![161715-21-5](/CAS/20180808/GIF/161715-21-5.gif)
Tebipenem Preparation Products And Raw materials
Raw materials
Preparation Products
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
career henan chemical co | +86-0371-86658258 +8613203830695 | sales@coreychem.com | China | 29901 | 58 |
Hubei Jusheng Technology Co.,Ltd. | 18871490254 | linda@hubeijusheng.com | CHINA | 28180 | 58 |
BOC Sciences | +1-631-485-4226 | inquiry@bocsci.com | United States | 19553 | 58 |
Chongqing Chemdad Co., Ltd | +86-023-6139-8061 +86-86-13650506873 | sales@chemdad.com | China | 39916 | 58 |
Neostar United (Changzhou) Industrial Co., Ltd. | +86-519-519-85557386 | marketing1@neostarunited.com | China | 12210 | 58 |
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | marketing@targetmol.com | United States | 19892 | 58 |
Shaanxi Dideu Medichem Co. Ltd | +86-029-89586680 +86-18192503167 | 1026@dideu.com | China | 9030 | 58 |
Baoji Guokang Bio-Technology Co., Ltd. | 0917-3909592 13892490616 | gksales1@gk-bio.com | China | 9326 | 58 |
Nanjing Doge Biomedical Technology Co., Ltd | +86-25-58227606 +86-15305155328 | sales@dogechemical.com | China | 4128 | 58 |
Wuhan Topule Biopharmaceutical Co., Ltd | +8618327326525 | masar@topule.com | China | 8474 | 58 |
View Lastest Price from Tebipenem manufacturers
Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
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2021-07-13 | Tebipenem
161715-21-5
|
US $15.00-10.00 / KG | 1KG | 99%+ HPLC | Monthly supply of 1 ton | Zhuozhou Wenxi import and Export Co., Ltd | |
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2021-07-10 | Tebipenem
161715-21-5
|
US $15.00-10.00 / KG | 1KG | 99%+ HPLC | Monthly supply of 1 ton | Zhuozhou Wenxi import and Export Co., Ltd | |
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2019-07-06 | Tebipenem
161715-21-5
|
US $1.00 / KG | 1G | 98% | 100KG | Career Henan Chemical Co |