(±)-ORG 28611

CAS No.
784138-08-5
Chemical Name:
(±)-ORG 28611
Synonyms
(±)-ORG 28611;[1-(cyclohexylmethyl)-7-methoxyindol-3-yl]-(3,4-dimethylpiperazin-1-yl)methanone
CBNumber:
CB63152409
Molecular Formula:
C23H33N3O2
Molecular Weight:
383.527
MDL Number:
MOL File:
784138-08-5.mol
Last updated:2023-04-23 13:52:06

(±)-ORG 28611 Properties

solubility DMF: 10 mg/ml; DMSO: 2 mg/ml; Ethanol: 20 mg/ml; Ethanol:PBS(pH 7.2) (1:1): 0.5 mg/ml
form A crystalline solid

(±)-ORG 28611 price More Price(6)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Cayman Chemical 15266 (±)-ORG 28611 ≥98% 784138-08-5 1mg $81 2024-03-01 Buy
Cayman Chemical 15266 (±)-ORG 28611 ≥98% 784138-08-5 5mg $356 2024-03-01 Buy
Cayman Chemical 15266 (±)-ORG 28611 ≥98% 784138-08-5 10mg $632 2024-03-01 Buy
TRC O671020 (±)-ORG28611 784138-08-5 5mg $290 2021-12-16 Buy
American Custom Chemicals Corporation API0028265 ORG-28611 95.00% 784138-08-5 5MG $458.84 2021-12-16 Buy
Product number Packaging Price Buy
15266 1mg $81 Buy
15266 5mg $356 Buy
15266 10mg $632 Buy
O671020 5mg $290 Buy
API0028265 5MG $458.84 Buy

(±)-ORG 28611 Chemical Properties,Uses,Production

Description

(±)-ORG 28611 is the racemic mixture of the water soluble, full agonist of the human cannabinoid (CB) receptors central CB1 (pEC50 = 7.6; pKi = 8.9) and peripheral CB2 (pKi = 8.8). ORG 28611 (0.1-1 μM/kg, intravenous) demonstrated antinociceptive activity in the mouse tail flick test and the mouse formalin paw test, and it was further evaluated clinically for use as a potential intravenous analgesic agent.

Uses

(±)-ORG 28611 is full agonist of the human cannabinoid (CB) receptors central CB1 (pEC50 = 7.6; pKi = 8.9) and peripheral CB2 (pKi = 8.8). ORG 28611 (0.1-1 μM/kg, intravenous) demonstrated antinociceptive activity in the mouse tail flick test and the mouse formalin paw test, and it was further evaluated clinically for use as a potential intravenous analgesic agent. Synthetic Cannabinoids

(±)-ORG 28611 Preparation Products And Raw materials

Raw materials

Preparation Products

(±)-ORG 28611 Suppliers

Global( 13)Suppliers
Supplier Tel Email Country ProdList Advantage
Shanghai Hongye Biotechnology Co. Ltd 400-9205774 sales@glpbio.cn China 6870 58
ChemeGen(Shanghai) Biotechnology Co.,Ltd. 18818260767 sales@chemegen.com China 11289 58
(±)-ORG 28611 [1-(cyclohexylmethyl)-7-methoxyindol-3-yl]-(3,4-dimethylpiperazin-1-yl)methanone 784138-08-5