(R)-3,4,5,6-tetrahydro-5-methyl-1-phenyl-1H-2,5-benzoxazocine hydrochloride
- CAS No.
- 53625-25-5
- Chemical Name:
- (R)-3,4,5,6-tetrahydro-5-methyl-1-phenyl-1H-2,5-benzoxazocine hydrochloride
- Synonyms
- (R)-nefopam hydrochloride;(R)-3,4,5,6-tetrahydro-5-methyl-1-phenyl-1H-2,5-benzoxazocine hydrochloride
- CBNumber:
- CB8931018
- Molecular Formula:
- C17H20ClNO
- Molecular Weight:
- 289.7998
- MDL Number:
- MOL File:
- 53625-25-5.mol
Last updated:2023-05-15 10:43:44
| solubility | DMSO (Slightly), Water (Slightly) |
|---|---|
| form | Solid |
| color | White to Off-White |
| FDA UNII | ZLW2D8CC3U |
(R)-3,4,5,6-tetrahydro-5-methyl-1-phenyl-1H-2,5-benzoxazocine hydrochloride Chemical Properties,Uses,Production
Uses
(-)-Nefopam inhibits the uptake of 5-hydroxytryptamine (5-HT), noradrenaline and dopamine in synaptosomal preparations from rat forebrain, hippocampus and striatum. A cyclized analog of orphenadrine and diphenhydramine; representative of a new class of centrally acting skeletal muscle relaxants, the benzoxazocines. Analgesic; antidepressant.
Definition
ChEBI: A hydrochloride obtained by reaction of (R)-nefopam with one equivalent of hydrochloric acid (the racemic salt is an analgesic drug).
(R)-3,4,5,6-tetrahydro-5-methyl-1-phenyl-1H-2,5-benzoxazocine hydrochloride Preparation Products And Raw materials
Raw materials
Preparation Products
(R)-3,4,5,6-tetrahydro-5-methyl-1-phenyl-1H-2,5-benzoxazocine hydrochloride
(R)-nefopam hydrochloride
53625-25-5