methylnaltrexone

methylnaltrexone Structure
CAS No.
83387-25-1
Chemical Name:
methylnaltrexone
Synonyms
Mrz 2663;Mrz-2663;Naltrexone mb;methylnaltrexone;Methylnaltrexonium;N-Methylnaltrexone;3-O-Methylnaltrexone;Naltrexone methyl ether;17-(Cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxymorphinanium-6-one;3-Methoxy-14-hydroxy-17-(cyclopropylmethyl)-4,5α-epoxymorphinan-6-one
CBNumber:
CB61314469
Molecular Formula:
C21H26NO4+
Molecular Weight:
356.43544
MOL File:
83387-25-1.mol
Modify Date:
2023/5/4 17:34:43

methylnaltrexone Chemical Properties,Uses,Production

General Description

Methylnaltrexone (Relistor) is the methylated, quaternaryform of naltrexone . The permanently chargednitrogen prevents the drug from crossing the blood-brainbarrier. Thus, it only acts as an antagonist at peripheralopioid receptors. Relistor was approved in April 2008 totreat opioid-induced constipation in patients receiving palliativecare. It is administered as a SC injection once everyother day.

methylnaltrexone Preparation Products And Raw materials

Raw materials

Preparation Products

Global( 3)Suppliers
Supplier Tel Country ProdList Advantage Inquiry
Pharmaffiliates Analytics and Synthetics P. Ltd +91-172-5066494 Haryana, India 6773 58 Inquiry
QUALITY CONTROL SOLUTIONS LTD. 13670046396 China 18865 58 Inquiry
TargetMol Chemicals Inc. 15002134094 China 28091 58 Inquiry

83387-25-1(methylnaltrexone)Related Search:

methylnaltrexone 17-(Cyclopropylmethyl)-4,5α-epoxy-3-methoxy-14-hydroxymorphinan-6-one 3-Methoxy-14-hydroxy-17-(cyclopropylmethyl)-4,5α-epoxymorphinan-6-one 3-O-Methylnaltrexone 4,5α-Epoxy-3-methoxy-14β-hydroxy-17-(cyclopropylmethyl)morphinan-6-one Naltrexone methyl ether 17-(Cyclopropylmethyl)-4,5alpha-epoxy-3,14-dihydroxy-17-methyl-6-oxomorphinanium 17-(Cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxymorphinanium-6-one Methylnaltrexonium Morphinanium, 17-(cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxy-17-methyl-6-oxo-, (5alpha)- Mrz 2663 Mrz-2663 Naltrexone mb N-Methylnaltrexone 83387-25-1