aprinocarsen 化学特性,用途語,生産方法
使用
Treatment of non-small
cell lung cancer (antisense oligonucleotide; protein kinase
C-alpha inhibitor).
brand name
Affinitak (Isis).
臨床応用
Aprinocarsen is a phosphorothioate antisense agent targeted against protein kinase Cα,
a protein that is implicated in malignant transformation and proliferation. It showed
activity in Phase I and Phase II clinical trials against nonsmall-cell lung cancer when
used in combination with cisplatin or the combination of cisplatin and gemcitabine.
aprinocarsen 上流と下流の製品情報
原材料
準備製品