PF-3274167 化学特性,用途語,生産方法
説明
PF-3274167 is an oxytocin receptor antagonist (K
i = 9.5 nM). It is selective for the oxytocin receptor over the vasopressin receptors V
1A and V
2 (K
is = 1,120 and 10,000 nM, respectively).
使用
PF-3274167 functions as s triazole oxytocin antagonists. It also functions as a PET radiotracer of oxytocin receptors.
PF-3274167 上流と下流の製品情報
原材料
準備製品