イメチット二臭化水素酸塩

イメチット二臭化水素酸塩 価格 もっと(4)

メーカー	製品番号	製品説明	CAS番号	包装	価格	更新時間	購入
富士フイルム和光純薬株式会社(wako)	W01TOC0729	イメチット二臭化水素酸塩 Imetit Dihydrobromide	32385-58-3	10mg	￥43000	2024-03-01	購入
富士フイルム和光純薬株式会社(wako)	W01TOC0729	イメチット二臭化水素酸塩 Imetit Dihydrobromide	32385-58-3	50mg	￥183000	2024-03-01	購入
Sigma-Aldrich Japan	I135	イメチット 二臭化水素酸塩 ≥98% (HPLC) Imetit dihydrobromide ≥98% (HPLC)	32385-58-3	10mg	￥20300	2024-03-01	購入
Sigma-Aldrich Japan	I135	イメチット 二臭化水素酸塩 ≥98% (HPLC) Imetit dihydrobromide ≥98% (HPLC)	32385-58-3	25mg	￥67100	2024-03-01	購入

イメチット二臭化水素酸塩 化学特性,用途語,生産方法

説明

Imetit is a histamine H₃ and H₄ receptor agonist (K_is = 0.3 and 2.7 nM, respectively, in radioligand binding assays). It is selective for histamine H₃ and H₄ receptors over H₁ and H₂ receptors at concentrations up to 100 μM, as well as the serotonin (5-HT) receptor subtype 5-HT₃ (K_i = 240 nM)., Imetit reduces potassium-induced increases in histamine levels in isolated rat cerebral cortex slices (EC₅₀ = 2.8 nM). It increases scratching in mice (ED₅₀ = 0.9 μmol), an effect that is reduced by the H₃ receptor antagonist thioperamide .

使用

Imetit dihydrobromide is a high affinity agonist at the histamine H3- and H4-receptors.

定義

ChEBI: A hydrobromide salt obtained by reaction of imetit with two equivalents of hydrobromic acid. An extremely potent, high affinity agonist at H3 and H4 receptors (Ki values are 0.3 and 2.7 nM respectively). Induces sh pe change in eosinophils with an EC50 of 25 nM. Centrally active following systemic administration.

生物活性

An extremely potent, high affinity agonist at H 3 and H 4 receptors (K i values are 0.3 and 2.7 nM respectively). Induces shape change in eosinophils with an EC 50 of 25 nM. Centrally active following systemic administration. Also available as part of the Histamine H 3 Receptor Tocriset™ .

イメチット二臭化水素酸塩 上流と下流の製品情報

原材料

準備製品

イメチット二臭化水素酸塩 生産企業

名前	電話番号	電子メール	国籍	製品カタログ	優位度
TargetMol Chemicals Inc.	+1-781-999-5354 +1-00000000000	marketing@targetmol.com	United States	19892	58
Hangzhou MolCore BioPharmatech Co.,Ltd.	+86-057181025280; +8617767106207	sales@molcore.com	China	49739	58
LEAPCHEM CO., LTD.	+86-852-30606658	market18@leapchem.com	China	43348	58
Aladdin Scientific	+1-+1(833)-552-7181	sales@aladdinsci.com	United States	57511	58
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
BOC Sciences	1-631-485-4226; 16314854226	info@bocsci.com	United States	14059	65
Hangzhou Sage Chemical Co., Ltd.	+86057186818502 13588463833	info@sagechem.com	China	10269	58
Sigma-Aldrich	021-61415566 800-8193336	orderCN@merckgroup.com	China	51471	80
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
Shanghai EFE Biological Technology Co., Ltd.	021-65675885 18964387627	info@efebio.com	China	9708	58

32385-58-3(イメチット二臭化水素酸塩)キーワード:

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• 32385-58-3
• S-[2-(IMIDAZOL-4-YL)ETHYL]ISOTHIOUREA DIHYDROBROMIDE
• 5-[2-(IMIDAZOL-4-YL)ETHYL]ISOTHIOUREA DIHYDROBROMIDE
• IMETIT DIHYDROBROMIDE
• IMETIT DIHYDROBROMIDE POTENT AND SELECTI VE
• S-[2-(Imidazol-4-yl)ethyl]isothiourea2HBr
• CarbaMiMidothioic acid, 2-(1H-iMidazol-4-yl)ethyl ester, dihydrobroMide
• S-[2-(4(5)-Imidazolyl)ethyl]isothiourea dihydrobromide
• SKF 91105 dihydrobromide
• VUF 8325 dihydrobromide
• Imetit dihydrobromid
• Imetit hydrobromide
• Carbamimidothioic acid, 2-(1H-imidazol-5-yl)ethyl ester, dihydrobromide
• イメチット二臭化水素酸塩
• イメチット 二臭化水素酸塩