Medetomidine hydrochloride 化学特性,用途語,生産方法
化学的特性
White to Off-White Crystalline Solid
使用
a2-Adrenergic aginist. Sedative; analgesic
生物活性
Potent, highly selective α 2 -adrenoceptor agonist (K i values are 1.08 and 1750 nM for α 2 - and α 1 -adrenoceptors respectively). Displays greater selectivity over α 1 -adrenoceptors than clonidine and UK 14,304 (1620-, 220- and 300-fold respectively). Inhibits twitch response in electrically stimulated mouse vas deferens (pD 2 = 9.0). Active in vivo ; displays hypotensive, bradycardic, sedative, anxiolytic, hypothermic and analgesic effects.
Medetomidine hydrochloride 上流と下流の製品情報
原材料
準備製品