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2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl-

2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl- 구조식 이미지

카스 번호:: 1010096-65-7

상품명:: 2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl-

동의어(영문):: AM6701;LY2183240 2’LY2183240 2’-isomer;LY2183240 2’-isomer Exclusive;LY2183240 2'-isomer Exclusive;5-([1,1-biphenyl]-4-ylmethyl)-N,N-dimethyl-2H-tetrazole-2-carboxamide;2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl-

CBNumber:: CB32667875

분자식:: C17H17N5O

포뮬러 무게:: 307.35

MOL 파일:: 1010096-65-7.mol

속성

안전

용도

공급 업체 11

2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl- 속성

끓는 점: 506.1±53.0 °C(Predicted)

밀도: 1.21±0.1 g/cm3(Predicted)

저장 조건: Store at -20°C

용해도: DMF: 3 mg/ml; DMSO: 2 mg/ml; Ethanol: 10 mg/ml; Ethanol:PBS(pH 7.2) (1:5): 0.1 mg/ml

물리적 상태: 결정성 고체

산도 계수 (pKa): -1.73±0.12(Predicted)

색상: Light yellow to yellow

안전

2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl- C화학적 특성, 용도, 생산

개요

LY2183240 is a potent, competitive small molecule inhibitor of anandamide uptake (IC₅₀ = 270 pM; K_i = 540 pM) and hydrolysis. It has been shown to increase anandamide levels in rat cerebellum (ED₅₀ = 1.37 mg/kg) and displays dose-dependent efficacy (3-30 mg/kg) in several rodent models of persistent pain. LY2183240 2’-isomer is a less potent, 2,5-regioisomer of LY2183240 that inhibits anandamide hydrolysis and uptake with IC₅₀ values of 33 and 998 nM, respectively.

용도

5-([1,1''-Biphenyl]-4-ylmethyl)-N,N-dimethyl-2H-tetrazole-2-carboxamide is an inhibitor of human monoacylglycerol lipase (hMGL).

2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl- 준비 용품 및 원자재

원자재

준비 용품

2H-Tetrazole-2-carboxaMide, 5-([1,1'-biphenyl]-4-ylMethyl)-N,N-diMethyl- 공급 업체

글로벌( 11)공급 업체

공급자	전화	이메일	국가	제품 수	이점
Haoyuan Chemexpress Co., Ltd.	021-58950125	info@chemexpress.com	China	7553	61
Shanghai Hongye Biotechnology Co. Ltd	400-9205774	sales@glpbio.cn	China	6870	58
BOC Sciences	--	info@bocsci.com	USA	0	65
Beijing Solarbio Science & Tecnology Co., Ltd.	010-50973130 17801761073	Gsiyu@solarbio.com	China	50471	58
Shanghai Yifei Biotechnology Co. , Ltd.	021-65675885 18964387627	customer_service@efebio.com	China	11975	58
https://hanhongsci.com/	021-54306202 18917919676	info@hanhongsci.com	China	29978	58