LAS101057
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LAS101057 속성
- 끓는 점
- 509.2±50.0 °C(Predicted)
- 밀도
- 1.400±0.06 g/cm3(Predicted)
- 저장 조건
- 2-8°C
- 용해도
- DMSO:125.0(Max Conc. mg/mL);372.75(Max Conc. mM)
- 물리적 상태
- 고체
- 산도 계수 (pKa)
- 11.70±0.20(Predicted)
- 색상
- White to off-white
안전
- 위험 및 안전 성명
- 위험 및 사전주의 사항 (GHS)
LAS101057 C화학적 특성, 용도, 생산
용도
LAS 101057 is a potent, selective, and orally efficacious A2B receptor antagonist, was identified as a clinical development candidate. It inhibits agonist-induced IL-6 production in human fibroblasts and is active in an ovalbumin (OVA)-sensitized mouse model after oral administration, reducing airway hyperresponsiveness to methacholine, Th2 cytokine production and OVA-specific IgE levels.LAS101057 준비 용품 및 원자재
원자재
준비 용품
LAS101057 공급 업체
글로벌( 20)공급 업체
공급자 | 전화 | 이메일 | 국가 | 제품 수 | 이점 |
---|---|---|---|---|---|
Fuxin Pharmaceutical | +86-021-021-50872116 +8613122107989 |
contact@fuxinpharm.com | China | 10297 | 58 |
TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 |
marketing@targetmol.com | United States | 19892 | 58 |
Jilin Chinese Academy of Sciences-yanshen Technology | +undefined18143011203 |
info@chemextension.com | China | 42057 | 58 |
Aladdin Scientific | +1-+1(833)-552-7181 |
sales@aladdinsci.com | United States | 52927 | 58 |
MedChemexpress LLC | 021-58955995 |
sales@medchemexpress.cn | United States | 4863 | 58 |
Shanghai Balmxy Pharmaceutical Co., Ltd | 021-24206007 13764915196 |
sales@balmxy.com | China | 6765 | 55 |
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd. | 025-66113011 18112977050 |
cb6@aikonchem.com | China | 16687 | 50 |
Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 |
info@efebio.com | China | 9806 | 58 |
Shanghai ZiHao Pharmaceutical Co., Ltd. | 021-13482410-12 13482410112 |
362383684@qq.com | China | 731 | 58 |
Cool Pharm, Ltd | 18019463053 |
sales@coolpharm.com | China | 13017 | 58 |