[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate
![[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate price.](/CAS/GIF/150080-09-4.gif)
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- $49 - $5127.15
- Product name: [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate
- CAS: 150080-09-4
- MF: C10H23BN2O6S
- MW: 310.17
- EINECS:
- MDL Number:MFCD13194906
- Synonyms:[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate;Boronic acid, ((2R)-1-((2S)-2-amino-3-methyl-1-oxobutyl)-2-pyrrolidinyl)-, monomethanesulfonate;Unii-V8zg4Y1B51;Methanesulfonic acid ((R)-1-((S)-2-amino-3-methyl-butanoyl)pyrrolidin-2-yl)boronic acid (1:1);Talabostat mesylate;Talabostat Mesilate;[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate Talabostat mesilate;Talabostat mesylate [(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate
31 prices
Selected condition：
Brand
- Adipogen Life Sciences
- American Custom Chemicals Corporation
- ApexBio Technology
- AvaChem
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 10
- 1mg
- 5mg
- 25mg
- 50
- 10mg
- 10mM(in 1mL DMSO)
- 50mg
- 100mg
- 250mg
- 1G
- ManufacturerAdipogen Life Sciences
- Product numberAG-CR1-3541-M050
- Product descriptionTalabostat.mesylate ≥98%(HPLC)
- Packaging50mg
- Price$220
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006399
- Product descriptionTALABOSTAT MESYLATE 95.00%
- Packaging1G
- Price$5127.15
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB3941
- Product descriptionTalabostatmesylate
- Packaging10mg
- Price$178
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB3941
- Product descriptionTalabostatmesylate
- Packaging10mM(in 1mL DMSO)
- Price$196
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2633
- Product descriptionTalabostat Mesylate
- Packaging5mg
- Price$105
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2633
- Product descriptionTalabostat Mesylate
- Packaging10mg
- Price$145
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2633
- Product descriptionTalabostat Mesylate
- Packaging25mg
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number2633
- Product descriptionTalabostat Mesylate
- Packaging100mg
- Price$545
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb546194
- Product descriptionTalabostat mesylate >98%
- Packaging10mg
- Price$173.4
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb546194
- Product descriptionTalabostat mesylate >98%
- Packaging50mg
- Price$447.1
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number29007
- Product descriptionTalabostat (mesylate)
- Packaging5mg
- Price$49
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29007
- Product descriptionTalabostat (mesylate)
- Packaging10mg
- Price$82
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29007
- Product descriptionTalabostat (mesylate)
- Packaging25mg
- Price$190
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29007
- Product descriptionTalabostat (mesylate)
- Packaging50mg
- Price$333
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-3187
- Product descriptionTalabostat(mesylate) 99.05%
- Packaging5mg
- Price$132
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-3187
- Product descriptionTalabostat(mesylate) 99.05%
- Packaging10mg
- Price$192
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Adipogen Life Sciences | AG-CR1-3541-M050 | Talabostat.mesylate ≥98%(HPLC) | 50mg | $220 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006399 | TALABOSTAT MESYLATE 95.00% | 1G | $5127.15 | 2021-12-16 | Buy |
| ApexBio Technology | B3941 | Talabostatmesylate | 10mg | $178 | 2021-12-16 | Buy |
| ApexBio Technology | B3941 | Talabostatmesylate | 10mM(in 1mL DMSO) | $196 | 2021-12-16 | Buy |
| AvaChem | 2633 | Talabostat Mesylate | 5mg | $105 | 2021-12-16 | Buy |
| AvaChem | 2633 | Talabostat Mesylate | 10mg | $145 | 2021-12-16 | Buy |
| AvaChem | 2633 | Talabostat Mesylate | 25mg | $245 | 2021-12-16 | Buy |
| AvaChem | 2633 | Talabostat Mesylate | 100mg | $545 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb546194 | Talabostat mesylate >98% | 10mg | $173.4 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb546194 | Talabostat mesylate >98% | 50mg | $447.1 | 2021-12-16 | Buy |
| Cayman Chemical | 29007 | Talabostat (mesylate) | 5mg | $49 | 2024-03-01 | Buy |
| Cayman Chemical | 29007 | Talabostat (mesylate) | 10mg | $82 | 2024-03-01 | Buy |
| Cayman Chemical | 29007 | Talabostat (mesylate) | 25mg | $190 | 2024-03-01 | Buy |
| Cayman Chemical | 29007 | Talabostat (mesylate) | 50mg | $333 | 2024-03-01 | Buy |
| ChemScene | CS-3187 | Talabostat(mesylate) 99.05% | 5mg | $132 | 2021-12-16 | Buy |
| ChemScene | CS-3187 | Talabostat(mesylate) 99.05% | 10mg | $192 | 2021-12-16 | Buy |
Properties
Melting point :>160°C (dec.)
storage temp. :under inert gas (nitrogen or Argon) at 2–8 °C
solubility :Soluble in DMSO (up to at least 25 mg/ml)
form :solid
color :White
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
storage temp. :under inert gas (nitrogen or Argon) at 2–8 °C
solubility :Soluble in DMSO (up to at least 25 mg/ml)
form :solid
color :White
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
Safety Information
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Description
Talabostat is a non-selective inhibitor of dipeptidyl peptidases (DPPs), including DPP-4, DPP-7, DPP-8, DPP-9, fibroblast activation protein (FAP), and prolyl endopeptidase (PREP; IC50s = >4, 310, 4, 11, 560, and 390 nM, respectively). It inhibits proliferation of superantigen-stimulated human peripheral blood mononuclear cells (PBMCs; IC50 = ~10 nM). Talabostat (5 μg twice per day) increases expression of a variety of cytokines, including those encoding IL-1β, IL-6, and G-CSF, and chemokines in tumors and tumor-draining lymph nodes in a WEHI-164 fibrosarcoma mouse model. It reduces tumor growth in WEHI-164, MM45T.Sp, and MM52.T fibrosarcoma, EL-4 and A20/2J lymphoma, B16/F10 melanoma, and P815 mastocytoma syngeneic mouse models. Talabostat also increases the efficacy of the antitumor antibodies rituximab and trastuzumab in Namalwa B cell lymphoma and LS180 colon carcinoma mouse xenograft models, respectively.Related product price
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Suppliers and manufacturers
career henan chemical co
![[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate](https://img.chemicalbook.com/ProductImageEN/2019-12/small/ab6cf7f8-e28f-44c5-9373-aaa3f286bf0d.jpg)
$6.60 /1KG
[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate CAS:150080-09-4
[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate CAS:150080-09-4
Dideu Industries Group Limited
![[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate](/ProductImageEN/2022-08/small/2c7d7b32-26c1-41c0-ab6e-52984d69cdec.jpg)
Alpha Biopharmaceuticals Co., Ltd
Capot Chemical Co.,Ltd.
ATK CHEMICAL COMPANY LIMITED
BOC Sciences
Chongqing Chemdad Co., Ltd
CONIER CHEM AND PHARMA LIMITED
Guangzhou Yuheng Pharmaceutical Technology Co., Ltd
WinWin Chemical CO., Limited
$1.10 /1g
[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate CAS:150080-09-4
[(2R)-1-[(2S)-2-Amino-3-methylbutanoyl]pyrrolidin-2-yl]boronic acid mesylate CAS:150080-09-4