L-Threonine, N-acetyl-L-threonyl-(αR)-α-hydroxybenzenepropanoyl-2,3-didehydro-N-methylalanyl-L-alanyl-N-methyl-L-alanyl-(3R)-3-[[(2S,3R)-2-(acetylamino)-3-hydroxy-4-methyl-1-oxopentyl]oxy]-L-leucyl-N,O-dimethyl-, (7→1)-lactone
- $250 - $370
- Product name: L-Threonine, N-acetyl-L-threonyl-(αR)-α-hydroxybenzenepropanoyl-2,3-didehydro-N-methylalanyl-L-alanyl-N-methyl-L-alanyl-(3R)-3-[[(2S,3R)-2-(acetylamino)-3-hydroxy-4-methyl-1-oxopentyl]oxy]-L-leucyl-N,O-dimethyl-, (7→1)-lactone
- CAS: 568580-02-9
- MF: C46H69N7O15
- MW: 960.09
- EINECS:
- MDL Number:MFCD09832722
- Synonyms:L-Threonine, N-acetyl-L-threonyl-(αR)-α-hydroxybenzenepropanoyl-2,3-didehydro-N-methylalanyl-L-alanyl-N-methyl-L-alanyl-(3R)-3-[[(2S,3R)-2-(acetylamino)-3-hydroxy-4-methyl-1-oxopentyl]oxy]-L-leucyl-N,O-dimethyl-, (7→1)-lactone
3 prices
Selected condition:
Brand
- Adipogen Life Sciences
- Cayman Chemical
- ChemScene
Package
- 250ug
- 1mg
- ManufacturerAdipogen Life Sciences
- Product numberAG-CN2-0509-M001
- Product descriptionYM-254890 ≥95%(HPLC)
- Packaging1mg
- Price$370
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number29735
- Product descriptionYM-254890
- Packaging1mg
- Price$335
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-0087171
- Product descriptionYM-254890 ≥99.0%
- Packaging250ug
- Price$250
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
Adipogen Life Sciences | AG-CN2-0509-M001 | YM-254890 ≥95%(HPLC) | 1mg | $370 | 2021-12-16 | Buy |
Cayman Chemical | 29735 | YM-254890 | 1mg | $335 | 2024-03-01 | Buy |
ChemScene | CS-0087171 | YM-254890 ≥99.0% | 250ug | $250 | 2021-12-16 | Buy |
Properties
Boiling point :1232.4±65.0 °C(Predicted)
Density :1.26±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :Soluble in DMSO (up to 10 mg/ml)
form :lyophilized solid
pka :12.52±0.70(Predicted)
color :White or off-white
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
Density :1.26±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :Soluble in DMSO (up to 10 mg/ml)
form :lyophilized solid
pka :12.52±0.70(Predicted)
color :White or off-white
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
Safety Information
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Description
YM-254890 (568580-02-9) is a novel Gαq/11 inhibitor.1 U46619-induced platelet aggregation is inhibited but phorbol ester- or ionophore-induced aggregation is not2 (IC50 = 0.1-0.2 μM)1. It blocks Pasteurella multocida toxin-mediated activation of Gαq.3 A highly useful new tool for studying Gαq/11-coupled receptor signaling and resulting cellular events.4Related product price
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