N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide
![N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide price.](/CAS/20150408/GIF/942206-85-1.gif)
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- $32 - $2700
- Product name: N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide
- CAS: 942206-85-1
- MF: C28H32Cl2N4O6S2
- MW: 655.61
- EINECS:
- MDL Number:MFCD12912413
- Synonyms:N-((S)-1-(4-((S)-2-(2,4-dichlorophenylsulfonaMido)-3-hydroxypropanoyl)piperazin-1-yl)-4-Methyl-1-oxopentan-2-yl)benzo[b]thiophene-2-carboxaMide;(N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide;GSK1016790A;GSK101;GSK1016790A;GSK-1016790A;GSK 1016790A;CS-2774;GSK-1016790A;GSK 1016790A;Benzo[b]thiophene-2-carboxamide, N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbonyl]-3-methylbutyl]-
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Brand
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Sigma-Aldrich
- Tocris
- TRC
Package
- 50
- 1MG
- 5mg
- 10MG
- 25mg
- 50MG
- 100mg
- 250mg
- 1g
- ManufacturerAK Scientific
- Product number0437DB
- Product descriptionGsk1016790A
- Packaging5mg
- Price$193
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0008289
- Product descriptionGSK1016790A 95.00%
- Packaging1MG
- Price$148.05
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0008289
- Product descriptionGSK1016790A 95.00%
- Packaging10MG
- Price$745.24
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0008289
- Product descriptionGSK1016790A 95.00%
- Packaging50MG
- Price$1297.64
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC5065
- Product descriptionGSK1016790A
- Packaging5mg
- Price$96
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC5065
- Product descriptionGSK1016790A
- Packaging10mg
- Price$158
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC5065
- Product descriptionGSK1016790A
- Packaging25mg
- Price$303
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number17289
- Product descriptionGSK1016790A ≥98%
- Packaging1mg
- Price$32
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17289
- Product descriptionGSK1016790A ≥98%
- Packaging5mg
- Price$86
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17289
- Product descriptionGSK1016790A ≥98%
- Packaging10mg
- Price$139
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17289
- Product descriptionGSK1016790A ≥98%
- Packaging25mg
- Price$267
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-5660
- Product descriptionGSK1016790A 99.67%
- Packaging5mg
- Price$84
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5660
- Product descriptionGSK1016790A 99.67%
- Packaging10mg
- Price$144
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5660
- Product descriptionGSK1016790A 99.67%
- Packaging25mg
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5660
- Product descriptionGSK1016790A 99.67%
- Packaging50mg
- Price$540
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5660
- Product descriptionGSK1016790A 99.67%
- Packaging100mg
- Price$900
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 0437DB | Gsk1016790A | 5mg | $193 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0008289 | GSK1016790A 95.00% | 1MG | $148.05 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0008289 | GSK1016790A 95.00% | 10MG | $745.24 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0008289 | GSK1016790A 95.00% | 50MG | $1297.64 | 2021-12-16 | Buy |
| ApexBio Technology | C5065 | GSK1016790A | 5mg | $96 | 2021-12-16 | Buy |
| ApexBio Technology | C5065 | GSK1016790A | 10mg | $158 | 2021-12-16 | Buy |
| ApexBio Technology | C5065 | GSK1016790A | 25mg | $303 | 2021-12-16 | Buy |
| Cayman Chemical | 17289 | GSK1016790A ≥98% | 1mg | $32 | 2024-03-01 | Buy |
| Cayman Chemical | 17289 | GSK1016790A ≥98% | 5mg | $86 | 2024-03-01 | Buy |
| Cayman Chemical | 17289 | GSK1016790A ≥98% | 10mg | $139 | 2024-03-01 | Buy |
| Cayman Chemical | 17289 | GSK1016790A ≥98% | 25mg | $267 | 2024-03-01 | Buy |
| ChemScene | CS-5660 | GSK1016790A 99.67% | 5mg | $84 | 2021-12-16 | Buy |
| ChemScene | CS-5660 | GSK1016790A 99.67% | 10mg | $144 | 2021-12-16 | Buy |
| ChemScene | CS-5660 | GSK1016790A 99.67% | 25mg | $300 | 2021-12-16 | Buy |
| ChemScene | CS-5660 | GSK1016790A 99.67% | 50mg | $540 | 2021-12-16 | Buy |
| ChemScene | CS-5660 | GSK1016790A 99.67% | 100mg | $900 | 2021-12-16 | Buy |
Properties
Melting point :>119°C (dec.)
Density :1.426±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: >10mg/mL
form :white solid
pka :8.29±0.50(Predicted)
color :White to Off-White
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
Density :1.426±0.06 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: >10mg/mL
form :white solid
pka :8.29±0.50(Predicted)
color :White to Off-White
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 2 months.
Safety Information
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Description
Transient receptor potential vanilloid 4 (TRPV4) is a nonselective cation channel thought to be involved in osmoregulation, hyperalgesia, and control of epithelial cell volume. GSK1016790A is a TRPV4 agonist that has been reported to elicit calcium influx in HEK cells expressing mouse or human TRPV4 (EC50s = 18 and 2.1 nM, respectively). It has been used to demonstrate a role for TRPV4 in regulating urinary bladder activity and endothelial control of vascular tone.More related product prices
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