GDC-0810(ARN-810)
|
- $36 - $1802
- Product name: GDC-0810(ARN-810)
- CAS: 1365888-06-7
- MF: C26H20ClFN2O2
- MW: 446.9
- EINECS:-0
- MDL Number:MFCD28902190
- Synonyms:(E)-3-(4-((E)-2-(2-CHLORO-4-FLUOROPHENYL)-1-(1H-INDAZOL-5-YL)BUT-1-EN-1-YL)PHENYL)ACRYLIC ACID;GDC-0810(ARN-810);GDC-0810;(E)-3-[4-[(E)-2-(2-Chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl]phenyl]-2-propenoic acid;GDC-0810 (Brilanestrant);ARN-810;ARN-810;BRILANESTRANT;CS-2080
20 prices
Selected condition：
Brand
- AK Scientific
- Biorbyt Ltd
- Biosynth Carbosynth
- Cayman Chemical
- Chemenu
- Crysdot
- DC Chemicals
- TRC
Package
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- ManufacturerAK Scientific
- Product number1882DN
- Product descriptionBrilanestrant
- Packaging100mg
- Price$1062
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb611604
- Product descriptionGDC-0810
- Packaging100mg
- Price$606.9
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb611604
- Product descriptionGDC-0810
- Packaging250mg
- Price$912.9
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb611604
- Product descriptionGDC-0810
- Packaging1g
- Price$1802
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFG137678
- Product descriptionGDC 0810
- Packaging5mg
- Price$100
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFG137678
- Product descriptionGDC 0810
- Packaging10mg
- Price$170
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFG137678
- Product descriptionGDC 0810
- Packaging25mg
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFG137678
- Product descriptionGDC 0810
- Packaging50mg
- Price$450
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFG137678
- Product descriptionGDC 0810
- Packaging100mg
- Price$750
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number29595
- Product descriptionARN810
- Packaging1mg
- Price$36
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29595
- Product descriptionARN810
- Packaging5mg
- Price$120
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29595
- Product descriptionARN810
- Packaging10mg
- Price$223
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29595
- Product descriptionARN810
- Packaging25mg
- Price$510
- Updated2024-03-01
- Buy
- ManufacturerChemenu
- Product numberCM295050
- Product description(E)-3-(4-((E)-2-(2-Chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl)phenyl)acrylicacid 98%
- Packaging50mg
- Price$1178
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31003730
- Product descriptionGDC-0810(ARN-810) 98+%
- Packaging10mg
- Price$285
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31003730
- Product descriptionGDC-0810(ARN-810) 98+%
- Packaging25mg
- Price$580
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 1882DN | Brilanestrant | 100mg | $1062 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb611604 | GDC-0810 | 100mg | $606.9 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb611604 | GDC-0810 | 250mg | $912.9 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb611604 | GDC-0810 | 1g | $1802 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FG137678 | GDC 0810 | 5mg | $100 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FG137678 | GDC 0810 | 10mg | $170 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FG137678 | GDC 0810 | 25mg | $300 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FG137678 | GDC 0810 | 50mg | $450 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FG137678 | GDC 0810 | 100mg | $750 | 2021-12-16 | Buy |
| Cayman Chemical | 29595 | ARN810 | 1mg | $36 | 2024-03-01 | Buy |
| Cayman Chemical | 29595 | ARN810 | 5mg | $120 | 2024-03-01 | Buy |
| Cayman Chemical | 29595 | ARN810 | 10mg | $223 | 2024-03-01 | Buy |
| Cayman Chemical | 29595 | ARN810 | 25mg | $510 | 2024-03-01 | Buy |
| Chemenu | CM295050 | (E)-3-(4-((E)-2-(2-Chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl)phenyl)acrylicacid 98% | 50mg | $1178 | 2021-12-16 | Buy |
| Crysdot | CD31003730 | GDC-0810(ARN-810) 98+% | 10mg | $285 | 2021-12-16 | Buy |
| Crysdot | CD31003730 | GDC-0810(ARN-810) 98+% | 25mg | $580 | 2021-12-16 | Buy |
Properties
Boiling point :622.8±55.0 °C(Predicted)
Density :1.342±0.06 g/cm3(Predicted)
solubility :DMSO:89.0(Max Conc. mg/mL);199.15(Max Conc. mM)
Ethanol:89.0(Max Conc. mg/mL);199.15(Max Conc. mM) form :A solid
pka :13.94±0.40(Predicted)
color :White to off-white
Density :1.342±0.06 g/cm3(Predicted)
solubility :DMSO:89.0(Max Conc. mg/mL);199.15(Max Conc. mM)
Ethanol:89.0(Max Conc. mg/mL);199.15(Max Conc. mM) form :A solid
pka :13.94±0.40(Predicted)
color :White to off-white
Safety Information
| Symbol(GHS): | ||||||||
|---|---|---|---|---|---|---|---|---|
| Signal word: | ||||||||
| Hazard statements: |
|
|||||||
| Precautionary statements: |
|
Description
Brilanestrant is an orally bioavailable Selective Estrogen Receptor Degrader (SERD) that demonstrates robust activity in tamoxifen-resistant breast cancer xenografts. GDC-0810 functions by binding to the estrogen receptor, inducing a conformational change resulting in the degradation of the receptor. GDC-0810 or ARN-810 demonstrates robust activity in models of tamoxifen-sensitive and tamoxifen-resistant breast cancer, and is currently in clinical trials in women with locally advanced or metastatic estrogen receptor-positive breast cancer.Related product price
- (-)-Varitriol
$1230 - Ethylamine
$10-1030.84 - ESTETROL
$35-2194.5
Suppliers and manufacturers
HANGZHOU CLAP TECHNOLOGY CO.,LTD
InvivoChem
Hangzhou MolCore BioPharmatech Co.,Ltd.
TargetMol Chemicals Inc.
Zibo Hangyu Biotechnology Development Co., Ltd
Aladdin Scientific
Amadis Chemical Company Limited
Shanghai Boyle Chemical Co., Ltd.
Chembest Research Laboratories Limited
WUHAN SUN-SHINE BIO-TECHNOLOGY Co., Ltd.