Lorediplon
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- $32 - $1500
- Product name: Lorediplon
- CAS: 917393-39-6
- MF: C20H15FN4O2S
- MW: 394.42
- EINECS:
- MDL Number:MFCD27987938
- Synonyms:Lorediplon;Thionorphine Hydrochloride;N-[2-fluoro-5-[3-(thiophene-2-carbonyl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl]-N-methylacetamide;Acetamide, N-[2-fluoro-5-[3-(2-thienylcarbonyl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl]-N-methyl-;GABA Receptor,γ-Aminobutyric acid Receptor,inhibit,Inhibitor,Lorediplon,Gamma-aminobutyric acid Receptor
13 prices
Selected condition：
Brand
- AK Scientific
- Cayman Chemical
- Chemenu
- ChemScene
- Crysdot
- DC Chemicals
Package
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- ManufacturerAK Scientific
- Product number2092CT
- Product descriptionLorediplon
- Packaging25mg
- Price$252
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number23868
- Product descriptionLorediplon ≥98%
- Packaging5mg
- Price$32
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number23868
- Product descriptionLorediplon ≥98%
- Packaging10mg
- Price$61
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number23868
- Product descriptionLorediplon ≥98%
- Packaging25mg
- Price$139
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number23868
- Product descriptionLorediplon ≥98%
- Packaging50mg
- Price$243
- Updated2024-03-01
- Buy
- ManufacturerChemenu
- Product numberCM255763
- Product descriptionN-(2-fluoro-5-(3-(thiophene-2-carbonyl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-N-methylacetamide 98%
- Packaging100mg
- Price$359
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5271
- Product descriptionLorediplon 99.78%
- Packaging10mg
- Price$50
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5271
- Product descriptionLorediplon 99.78%
- Packaging50mg
- Price$200
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000266
- Product descriptionLorediplon 98+%
- Packaging50mg
- Price$329
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000266
- Product descriptionLorediplon 98+%
- Packaging100mg
- Price$534
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC8642
- Product descriptionLorediplon >98%
- Packaging100mg
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC8642
- Product descriptionLorediplon >98%
- Packaging250mg
- Price$600
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC8642
- Product descriptionLorediplon >98%
- Packaging1g
- Price$1500
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 2092CT | Lorediplon | 25mg | $252 | 2021-12-16 | Buy |
| Cayman Chemical | 23868 | Lorediplon ≥98% | 5mg | $32 | 2024-03-01 | Buy |
| Cayman Chemical | 23868 | Lorediplon ≥98% | 10mg | $61 | 2024-03-01 | Buy |
| Cayman Chemical | 23868 | Lorediplon ≥98% | 25mg | $139 | 2024-03-01 | Buy |
| Cayman Chemical | 23868 | Lorediplon ≥98% | 50mg | $243 | 2024-03-01 | Buy |
| Chemenu | CM255763 | N-(2-fluoro-5-(3-(thiophene-2-carbonyl)pyrazolo[1,5-a]pyrimidin-7-yl)phenyl)-N-methylacetamide 98% | 100mg | $359 | 2021-12-16 | Buy |
| ChemScene | CS-5271 | Lorediplon 99.78% | 10mg | $50 | 2021-12-16 | Buy |
| ChemScene | CS-5271 | Lorediplon 99.78% | 50mg | $200 | 2021-12-16 | Buy |
| Crysdot | CD31000266 | Lorediplon 98+% | 50mg | $329 | 2021-12-16 | Buy |
| Crysdot | CD31000266 | Lorediplon 98+% | 100mg | $534 | 2021-12-16 | Buy |
| DC Chemicals | DC8642 | Lorediplon >98% | 100mg | $300 | 2021-12-16 | Buy |
| DC Chemicals | DC8642 | Lorediplon >98% | 250mg | $600 | 2021-12-16 | Buy |
| DC Chemicals | DC8642 | Lorediplon >98% | 1g | $1500 | 2021-12-16 | Buy |
Properties
storage temp. :Store at -20°C
solubility :DMF: 25 mg/ml; DMF:PBS(pH 7.2)(1:1): 0.5 mg/ml; DMSO: 14 mg/ml
form :A crystalline solid
color :Light yellow to yellow
solubility :DMF: 25 mg/ml; DMF:PBS(pH 7.2)(1:1): 0.5 mg/ml; DMSO: 14 mg/ml
form :A crystalline solid
color :Light yellow to yellow
Safety Information
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Description
Lorediplon is a non-benzodiazepine belonging to pyrazolopyrimidine family isunderdevelopment for the management for insomnia. Lorediplon acts by modulationof the GABAgreceptor. Its long plasma half-life has the potential of hypnotic effect. Ithas the potential for maintenance of sleep and the sleep architecture. In the phase Ipharmacodynamic study,it showed better efficacy in quality and maintenance ofsleep as compared with zolpidem. It has been shown to be well tolerated, safe with noresidual effects as compared with other sedative-hypnotic. Currently, the drug has completed Phase ll clinical trial. Results indicated strongefficacy in sleep maintenance with an acceptable safety profile. It also seems topreserve natural sleep architecture.Suppliers and manufacturers
ATK CHEMICAL COMPANY LIMITED
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SHANGHAI KEAN TECHNOLOGY CO., LTD.
Amadis Chemical Company Limited
Haoyuan Chemexpress Co., Ltd.
MedChemexpress LLC
