Mirogabalin
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- $68 - $3500
- Product name: Mirogabalin
- CAS: 1138245-13-2
- MF: C12H19NO2
- MW: 209.28
- EINECS:-0
- MDL Number:MFCD28411425
- Synonyms:Mirogabalin;[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid;A200-0700;DS5565;A200-0700;2-[(1R,5S,6S)-6-(aminomethyl)-3-ethyl-6-bicyclo[3.2.0]hept-3-enyl]acetic acid;MIROGABALIN; DS-5565;DS 5565;DS-5565;DS5565;Bicyclo[3.2.0]hept-3-ene-6-acetic acid, 6-(aminomethyl)-3-ethyl-, (1R,5S,6S)-
17 prices
Selected condition：
Brand
- AK Scientific
- American Custom Chemicals Corporation
- Biosynth Carbosynth
- Cayman Chemical
- Chemenu
- ChemScene
- DC Chemicals
- TRC
Package
- 1mg
- 2.5mg
- 5MG
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- 100g
- ManufacturerAK Scientific
- Product number4972DP
- Product descriptionMirogabalin
- Packaging10mg
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0028663
- Product descriptionMIROGABALIN 95.00%
- Packaging5MG
- Price$496.06
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBM166964
- Product descriptionMirogabalin
- Packaging10mg
- Price$145
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBM166964
- Product descriptionMirogabalin
- Packaging50mg
- Price$507.5
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number22475
- Product descriptionMirogabalin ≥98%
- Packaging1mg
- Price$68
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number22475
- Product descriptionMirogabalin ≥98%
- Packaging5mg
- Price$152
- Updated2024-03-01
- Buy
- ManufacturerChemenu
- Product numberCM247838
- Product descriptionMirogabalin 98%
- Packaging100g
- Price$3500
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging5mg
- Price$120
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging10mg
- Price$190
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging25mg
- Price$300
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging50mg
- Price$450
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-6008
- Product descriptionMirogabalin 99.31%
- Packaging100mg
- Price$750
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC10013
- Product descriptionMirogabalin >98%
- Packaging100mg
- Price$700
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC10013
- Product descriptionMirogabalin >98%
- Packaging250mg
- Price$1300
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC10013
- Product descriptionMirogabalin >98%
- Packaging1g
- Price$2500
- Updated2021-12-16
- Buy
- ManufacturerTRC
- Product numberM364940
- Product descriptionMirogabalin
- Packaging1mg
- Price$140
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 4972DP | Mirogabalin | 10mg | $245 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0028663 | MIROGABALIN 95.00% | 5MG | $496.06 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BM166964 | Mirogabalin | 10mg | $145 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BM166964 | Mirogabalin | 50mg | $507.5 | 2021-12-16 | Buy |
| Cayman Chemical | 22475 | Mirogabalin ≥98% | 1mg | $68 | 2024-03-01 | Buy |
| Cayman Chemical | 22475 | Mirogabalin ≥98% | 5mg | $152 | 2024-03-01 | Buy |
| Chemenu | CM247838 | Mirogabalin 98% | 100g | $3500 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 5mg | $120 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 10mg | $190 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 25mg | $300 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 50mg | $450 | 2021-12-16 | Buy |
| ChemScene | CS-6008 | Mirogabalin 99.31% | 100mg | $750 | 2021-12-16 | Buy |
| DC Chemicals | DC10013 | Mirogabalin >98% | 100mg | $700 | 2021-12-16 | Buy |
| DC Chemicals | DC10013 | Mirogabalin >98% | 250mg | $1300 | 2021-12-16 | Buy |
| DC Chemicals | DC10013 | Mirogabalin >98% | 1g | $2500 | 2021-12-16 | Buy |
| TRC | M364940 | Mirogabalin | 1mg | $140 | 2021-12-16 | Buy |
Properties
Boiling point :357.5±15.0 °C(Predicted)
Density :1.104±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF:0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Ethanol:1.25(Max Conc. mg/mL);5.97(Max Conc. mM)
PBS (pH 7.2):0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Water:5.36(Max Conc. mg/mL);25.61(Max Conc. mM) form :A crystalline solid
pka :4.65±0.10(Predicted)
color :Light yellow to light brown
InChI :InChI=1S/C12H19NO2/c1-2-8-3-9-5-12(7-13,6-11(14)15)10(9)4-8/h4,9-10H,2-3,5-7,13H2,1H3,(H,14,15)/t9-,10-,12-/m1/s1
InChIKey :FTBQORVNHOIASH-CKYFFXLPSA-N
SMILES :[C@]12([H])[C@]([H])([C@@](CN)(CC(O)=O)C1)C=C(CC)C2
Density :1.104±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF:0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Ethanol:1.25(Max Conc. mg/mL);5.97(Max Conc. mM)
PBS (pH 7.2):0.5(Max Conc. mg/mL);2.39(Max Conc. mM)
Water:5.36(Max Conc. mg/mL);25.61(Max Conc. mM) form :A crystalline solid
pka :4.65±0.10(Predicted)
color :Light yellow to light brown
InChI :InChI=1S/C12H19NO2/c1-2-8-3-9-5-12(7-13,6-11(14)15)10(9)4-8/h4,9-10H,2-3,5-7,13H2,1H3,(H,14,15)/t9-,10-,12-/m1/s1
InChIKey :FTBQORVNHOIASH-CKYFFXLPSA-N
SMILES :[C@]12([H])[C@]([H])([C@@](CN)(CC(O)=O)C1)C=C(CC)C2
Safety Information
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Description
Mirogabalin is a calcium channel blocker with analgesic effects. It binds to the α2δ-1 and α2δ-2 subunits of voltage-dependent Ca2+ channels. Mirogabalin has potent and sustained analgesic effects (ED50 = 2.5 mg/kg) in rats with diabetes induced by streptozotocin (STZ; ). Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID50 = 9.4 mg/kg) or locomotor activity (ID50 = 43.9 mg/kg), at its effective dose. Formulations containing mirogabalin are in clinical trials for diabetic peripheral neuropathic pain.Suppliers and manufacturers
Beijing Hope Pharmaceutical Co., Ltd.
ATK CHEMICAL COMPANY LIMITED
BOC Sciences
HANGZHOU CLAP TECHNOLOGY CO.,LTD
AFINE CHEMICALS LIMITED
Finetech Industry Limited
Zhejiang J&C Biological Technology Co.,Limited
