PD 168077 MALEATE
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- $93 - $5053
- Product name: PD 168077 MALEATE
- CAS: 630117-19-0
- MF: C24H26N4O5
- MW: 450.49
- EINECS:
- MDL Number:MFCD01321067
- Synonyms:N-(METHYL-4-(2-CYANOPHENYL)PIPERAZINYL)-3-METHYLBENZAMIDE MALEATE;PD 168077 MALEATE;N-[[4-(2-CYANOPHENYL)-1-PIPERAZINYL]METHYL]-3-METHYL-BENZAMIDE MALEATE;PD 168077 (maL;Benzamide,N-[[4-(2-cyanophenyl)-1-piperazinyl]methyl]-3-methyl-,(2Z)-2-butenedioate(1:1);PD 168077,Dopamine Receptor,PD-168077,inhibit,PD168077,PD168077 maleate,Inhibitor,PD 168077 maleate
28 prices
Selected condition：
Brand
- Ambeed
- ApexBio Technology
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- DC Chemicals
- Sigma-Aldrich
- Tocris
- Usbiological
Package
- 50
- 5mg
- 10
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- ManufacturerAmbeed
- Product numberA447591
- Product descriptionN-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+%
- Packaging5mg
- Price$285
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA447591
- Product descriptionN-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+%
- Packaging10mg
- Price$370
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA447591
- Product descriptionN-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+%
- Packaging25mg
- Price$480
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA447591
- Product descriptionN-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+%
- Packaging50mg
- Price$624
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA447591
- Product descriptionN-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+%
- Packaging100mg
- Price$810
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA447591
- Product descriptionN-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+%
- Packaging1g
- Price$5053
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6578
- Product descriptionPD168077maleate
- Packaging5mg
- Price$158
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6578
- Product descriptionPD168077maleate
- Packaging10mg
- Price$236
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6578
- Product descriptionPD168077maleate
- Packaging25mg
- Price$488
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6578
- Product descriptionPD168077maleate
- Packaging50mg
- Price$819
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6578
- Product descriptionPD168077maleate
- Packaging100mg
- Price$1386
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb572969
- Product descriptionPD-168077 maleate >98%
- Packaging100mg
- Price$838.1
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb572969
- Product descriptionPD-168077 maleate >98%
- Packaging250mg
- Price$1654.1
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb572969
- Product descriptionPD-168077 maleate >98%
- Packaging1g
- Price$3282.7
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number29789
- Product descriptionPD 168077 (maleate)
- Packaging5mg
- Price$93
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29789
- Product descriptionPD 168077 (maleate)
- Packaging10mg
- Price$166
- Updated2024-03-01
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Ambeed | A447591 | N-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+% | 5mg | $285 | 2021-12-16 | Buy |
| Ambeed | A447591 | N-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+% | 10mg | $370 | 2021-12-16 | Buy |
| Ambeed | A447591 | N-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+% | 25mg | $480 | 2021-12-16 | Buy |
| Ambeed | A447591 | N-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+% | 50mg | $624 | 2021-12-16 | Buy |
| Ambeed | A447591 | N-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+% | 100mg | $810 | 2021-12-16 | Buy |
| Ambeed | A447591 | N-((4-(2-Cyanophenyl)piperazin-1-yl)methyl)-3-methylbenzamidemaleate 95+% | 1g | $5053 | 2021-12-16 | Buy |
| ApexBio Technology | B6578 | PD168077maleate | 5mg | $158 | 2021-12-16 | Buy |
| ApexBio Technology | B6578 | PD168077maleate | 10mg | $236 | 2021-12-16 | Buy |
| ApexBio Technology | B6578 | PD168077maleate | 25mg | $488 | 2021-12-16 | Buy |
| ApexBio Technology | B6578 | PD168077maleate | 50mg | $819 | 2021-12-16 | Buy |
| ApexBio Technology | B6578 | PD168077maleate | 100mg | $1386 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb572969 | PD-168077 maleate >98% | 100mg | $838.1 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb572969 | PD-168077 maleate >98% | 250mg | $1654.1 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb572969 | PD-168077 maleate >98% | 1g | $3282.7 | 2021-12-16 | Buy |
| Cayman Chemical | 29789 | PD 168077 (maleate) | 5mg | $93 | 2024-03-01 | Buy |
| Cayman Chemical | 29789 | PD 168077 (maleate) | 10mg | $166 | 2024-03-01 | Buy |
Properties
storage temp. :Inert atmosphere,2-8°C
solubility :DMSO: >10 mg/mL
form :powder
color :white
solubility :DMSO: >10 mg/mL
form :powder
color :white
Safety Information
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| Signal word: | Warning | ||||||||||||||
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Description
PD 168077 is a dopamine D4 receptor agonist (Ki = 8.7 nM in CHO Pro 5 cells expressing the human receptor). It is selective for dopamine D4 over D2 and D3 receptors (Kis = 3,740 and 2,810 nM, respectively), as well as α1- and α2-adrenergic and serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT2A (Kis = 168, 177, 385, and 4,010 nM, respectively). PD 168077 (20 μM) induces CaMKII translocation from the dendritic shaft to postsynaptic sites on the dendritic processes of primary rat embryonic prefrontal cortex pyramidal neurons, an effect that can be blocked by the IP3 receptor antagonist 2APB or the calcium chelator BAPTA AM . PD 168077 (50-200 ng/animal) induces penile erections in rats when injected into the paraventricular nucleus (PVN) of the hypothalamus. PD 168077 (0.2-25 mg/kg, s.c.) increases spontaneous locomotor activity and reduces grooming and rearing in rats.Suppliers and manufacturers
ATK CHEMICAL COMPANY LIMITED
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3B Pharmachem (Wuhan) International Co.,Ltd.
EMMX Biotechnology LLC
Shanghai EFE Biological Technology Co., Ltd.