PICROTIN
- $32 - $733.72
- Product name: PICROTIN
- CAS: 21416-53-5
- MF: C15H18O7
- MW: 310.3
- EINECS:
- MDL Number:MFCD00868514
- Synonyms:PICROTIN;(1aR,8aS,9S)-1aβ,2,2a,6,6aα,8b-Hexahydro-2aα-hydroxy-9-(1-hydroxy-1-methylethyl)-8bα-methyl-3α,6α-methano-8H-1,5,7-trioxacyclopenta[ij]cycloprop[a]azulene-4,8(3H)-dione;(1aR,2aR,3S,6R,6aS,8aS,8bR,9S)-Hexahydro-2a-hydroxy-9-(1-hydroxy-1-methylethyl)-8b-methyl-3,6-methano-8H-1,5,7-trioxacyclopenta[ij]cycloprop[a]azulene-4,8(3H)-dione;Picrotin CRS;3,6-Methano-8H-1,5,7-trioxacyclopenta[ij]cycloprop[a]azulene-4,8(3H)-dione, hexahydro-2a-hydroxy-9-(1-hydroxy-1-methylethyl)-8b-methyl-, (1aR,2aR,3S,6R,6aS,8aS,8bR,9S)-
11 prices
Selected condition:
Brand
- American Custom Chemicals Corporation
- Biosynth Carbosynth
- Cayman Chemical
- Sigma-Aldrich
- TRC
Package
- 50mg
- 100mg
- 25mg
- y0001508
- 250MG
- 500mg
- 1G
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberCHM0031808
- Product descriptionPICROTIN 95.00%
- Packaging250MG
- Price$603.95
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberCHM0031808
- Product descriptionPICROTIN 95.00%
- Packaging1G
- Price$733.72
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFP66559
- Product descriptionPicrotin
- Packaging250mg
- Price$70
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFP66559
- Product descriptionPicrotin
- Packaging500mg
- Price$112.5
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFP66559
- Product descriptionPicrotin
- Packaging1g
- Price$180
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number21870
- Product descriptionPicrotin ≥98%
- Packaging25mg
- Price$32
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21870
- Product descriptionPicrotin ≥98%
- Packaging50mg
- Price$57
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21870
- Product descriptionPicrotin ≥98%
- Packaging100mg
- Price$98
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21870
- Product descriptionPicrotin ≥98%
- Packaging250mg
- Price$169
- Updated2024-03-01
- Buy
- ManufacturerSigma-Aldrich
- Product numberY0001508
- Product descriptionPicrotin European Pharmacopoeia (EP) Reference Standard
- Packagingy0001508
- Price$220
- Updated2024-03-01
- Buy
- ManufacturerTRC
- Product numberP437638
- Product descriptionPicrotin
- Packaging50mg
- Price$90
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
American Custom Chemicals Corporation | CHM0031808 | PICROTIN 95.00% | 250MG | $603.95 | 2021-12-16 | Buy |
American Custom Chemicals Corporation | CHM0031808 | PICROTIN 95.00% | 1G | $733.72 | 2021-12-16 | Buy |
Biosynth Carbosynth | FP66559 | Picrotin | 250mg | $70 | 2021-12-16 | Buy |
Biosynth Carbosynth | FP66559 | Picrotin | 500mg | $112.5 | 2021-12-16 | Buy |
Biosynth Carbosynth | FP66559 | Picrotin | 1g | $180 | 2021-12-16 | Buy |
Cayman Chemical | 21870 | Picrotin ≥98% | 25mg | $32 | 2024-03-01 | Buy |
Cayman Chemical | 21870 | Picrotin ≥98% | 50mg | $57 | 2024-03-01 | Buy |
Cayman Chemical | 21870 | Picrotin ≥98% | 100mg | $98 | 2024-03-01 | Buy |
Cayman Chemical | 21870 | Picrotin ≥98% | 250mg | $169 | 2024-03-01 | Buy |
Sigma-Aldrich | Y0001508 | Picrotin European Pharmacopoeia (EP) Reference Standard | y0001508 | $220 | 2024-03-01 | Buy |
TRC | P437638 | Picrotin | 50mg | $90 | 2021-12-16 | Buy |
Properties
Melting point :256-258°C
alpha :D -64.7° (c = 2.31 in abs alc)
Boiling point :595.8±50.0 °C(Predicted)
Density :1.59
storage temp. :2-8°C
solubility :DMF: 30 mg/ml; DMSO: 30 mg/ml; DMSO:PBS (pH 7.2)(1:9): 0.1 mg/ml
pka :13.28±0.60(Predicted)
form :Solid
color :White to off-white
EPA Substance Registry System :Picrotin (21416-53-5)
alpha :D -64.7° (c = 2.31 in abs alc)
Boiling point :595.8±50.0 °C(Predicted)
Density :1.59
storage temp. :2-8°C
solubility :DMF: 30 mg/ml; DMSO: 30 mg/ml; DMSO:PBS (pH 7.2)(1:9): 0.1 mg/ml
pka :13.28±0.60(Predicted)
form :Solid
color :White to off-white
EPA Substance Registry System :Picrotin (21416-53-5)
Safety Information
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Description
Picrotin is a natural picrotoxane that antagonizes glycine receptors (GlyRs; IC50s = 57 and 117 μM for α1 and α2 homodimeric GlyRs, respectively). It also inhibits α3 homodimeric GlyRs. Picrotin is inactive in inhibiting γ-aminobutyric acid (GABA) type A and type C receptors. Picrotin occurs in the natural plant-derived poison picrotoxin , equimolar with picrotoxinin.More related product prices
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