| | 143322-58-1 Basic information More.. |
| Product Name: | Eletriptan | | Synonyms: | ELETRIPTAN;3-[(1-methylpyrrolidin-2-yl)methyl]-5-(2-phenylsulfonylethyl)-1h-indole;5-(2-(Benzenesulfoyl)vinyl)-3-(1-Methylpyrrolidin-2(R)-ylmethyl)-1H-Indole;EletriptanHydrobromide(ForR&DOnly);UK-116044,Relpax,3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole;5-(2-(BENZENESULFONYL)VINYL)-3-(1-METHYLPYRROLIDIN-2(R)-YLMETHYL)-1H-INDOLE;3-[[(R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]indolemonohydrobromide;3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole | | CAS: | 143322-58-1 | | MF: | C22H26N2O2S | | MW: | 382.52 | | EINECS: | | | Mol File: | 143322-58-1.mol |  |
Use
Eletriptan is a 5-ht receptor agonist that binds to 5-ht1b, 5ht1d and 5ht1f receptors with high potency. activation of these receptors causes constriction of extracerebral intracranial vessels, abolition of the dural extravasation and neurogenic inflammation, and inhibition of trigeminal neuronal discharge. eletriptan was found to be the most potent agonist at the 5-ht1d receptor compared to the other triptans with pec50 value of 9.2.
- Eletriptan
-
- US $200.00 / kg
- 2023-06-26
- CAS:143322-58-1
- Min. Order: 1kg
- Purity: 99%
- Supply Ability: 1000kg/Month
- eletriptan
-
- US $150.00 / kg
- 2023-05-27
- CAS:143322-58-1
- Min. Order: 1kg
- Purity: 99.9%
- Supply Ability: 10000MT
- Eletriptan
-
- US $100.00 / g
- 2023-04-11
- CAS:143322-58-1
- Min. Order: 10g
- Purity: 99%
- Supply Ability: 1000g
|
|
143322-58-1
Recommend Suppliers |
|