| 169528-11-4 Basic information More.. |
Product Name: | PD-149163 | Synonyms: | PD-149163;L-Leucine, N2-[(2S)-2,6-diaminohexyl]-L-lysyl-L-prolyl-L-tryptophyl-3-methyl-L-valyl-, ethyl ester | CAS: | 169528-11-4 | MF: | C42H71N9O6 | MW: | 798.07 | EINECS: | | Mol File: | 169528-11-4.mol | |
Use
PD 149163 is a selective, brain penetrating Neurotensin NTR1 receptor agonist. Neurotensin agonists such as PD 149163 block the prepulse inhibition deficits produced by a 5-HT2A and an α1 agonist. As a result, PD 149163 shows pro-cognitive, antipsychotic and anxiolytic effects.
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169528-11-4
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