169528-11-4 Basic information More..
Product Name:PD-149163
Synonyms:PD-149163;L-Leucine, N2-[(2S)-2,6-diaminohexyl]-L-lysyl-L-prolyl-L-tryptophyl-3-methyl-L-valyl-, ethyl ester
CAS:169528-11-4
MF:C42H71N9O6
MW:798.07
EINECS:
Mol File:169528-11-4.mol
169528-11-4

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PD 149163 is a selective, brain penetrating Neurotensin NTR1 receptor agonist. Neurotensin agonists such as PD 149163 block the prepulse inhibition deficits produced by a 5-HT2A and an α1 agonist. As a result, PD 149163 shows pro-cognitive, antipsychotic and anxiolytic effects.

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