| 1197160-78-3 Basic information More.. |
Product Name: | PF-05212384 | Synonyms: | PF-05212384;PKI587;N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]phenyl]urea;1-(4-(4-(dimethylamino)piperidine-1-carbonyl)phenyl)-3-(4-(4,6-dimorpholino-1,3,5-triazin-2-yl)phenyl)urea;Gedatolisib (PF-05212384, PKI-587);N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]phenyl]urea PF-05212384 (PKI-587);PKI-587 N-[4-[[4-(Dimethylamino)-1-piperidinyl]carbonyl]phenyl]-N'-[4-[4,6-di(4-morpholinyl)-1,3,5-triazin-2-yl]phenyl]urea;PKI-587 ( Gedatolisib ) | CAS: | 1197160-78-3 | MF: | C32H41N9O4 | MW: | 615.73 | EINECS: | | Mol File: | 1197160-78-3.mol | |
Use
Gedatolisib (PF-05212384, PKI-587) is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC50 of 0.4 nM, 5.4 nM and 1.6 nM in cell-free assays, respectively. Phase 2.
- Gedatolisib;PKI-587
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- US $200.00-0.00 / g
- 2021-10-08
- CAS:1197160-78-3
- Min. Order: 1g
- Purity: 98%+
- Supply Ability: 100kgs
- PF-05212384
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- US $2.00 / kg
- 2019-07-06
- CAS:1197160-78-3
- Min. Order: 1kg
- Purity: 99%
- Supply Ability: 100kg
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1197160-78-3
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