1208222-39-2 Basic information More..
Product Name:VU 0365114
Synonyms:VU 0365114;1-Biphenyl-4-ylmethyl-5-trifluoromethoxy-1H-indole-2,3-dione;1-[(1,1'-Biphenyl)-4-ylmethyl]-5-(trifluoromethoxy)-1H-indole-2,3-dione;1H-Indole-2,3-dione, 1-([1,1'-biphenyl]-4-ylmethyl)-5-(trifluoromethoxy)-;VU 0365114,inhibit,Muscarinic acetylcholine receptor,VU0365114,Inhibitor,VU-0365114,mAChR;1-([1,1'-Biphenyl]-4-ylmethyl)-5-(trifluoromethoxy)indoline-2,3-dione
CAS:1208222-39-2
MF:C22H14F3NO3
MW:397.35
EINECS:
Mol File:1208222-39-2.mol
1208222-39-2

Use

VU 0365114 is a selective positive allosteric modulator of M5 (EC50 values are 2.7 μM for human M5, and >30 μM for M1, M2, M3 and M4 receptors).

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