| Company Name: |
Shanghai Yifei Biotechnology Co. , Ltd.
|
| Tel: |
021-65675885 18964387627 |
| Email: |
customer_service@efebio.com |
| Products Intro: |
Product Name:(Rac)-CP-601927 hydrochloride
CAS:230615-01-7
Purity:95% Package:2mg
|
| Company Name: |
TargetMol Chemicals Inc.
|
| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:(Rac)-CP-601927 hydrochloride
CAS:230615-01-7
Package:2mg/RMB 2120
|
|
| | (Rac)-CP-601927 hydrochloride Basic information |
| | (Rac)-CP-601927 hydrochloride Chemical Properties |
| storage temp. | 4°C, away from moisture | | form | Solid | | color | Off-white to light yellow |
| | (Rac)-CP-601927 hydrochloride Usage And Synthesis |
| Biological Activity | (Rac)-CP-601927 hydrochloride is the racemate of CP-601927. CP-601927 is a nAChR agonist with Ki values 1.2 nM and 102 nM for α4β2 and α3β4 nAChR, respectively[1].
CP-601927 induces significant antidepressant-like effects in mice. CP-601927 could decrease cholinergic signaling as a result of its reduced efficacy or via desensitization of α4β2* nAChRs[1]. | | References | [1]. Yann S Mineur, et al. α4β2 nicotinic acetylcholine receptor partial agonists with low intrinsic efficacy have antidepressant-like properties. Behav Pharmacol. 2011 Aug;22(4):291-9. |
| | (Rac)-CP-601927 hydrochloride Preparation Products And Raw materials |
|