ERK2/p38α MAPK-IN-1

Request For Quotation

ERK2/p38α MAPK-IN-1 Suppliers list

Company Name:	TargetMol Chemicals Inc.
Tel:	15002134094
Email:	marketing@targetmol.cn
Products Intro:	Product Name:ERK2/p38α MAPK-IN-1 CAS:1016427-72-7 Package:10mg;50mg

ERK2/p38α MAPK-IN-1 Basic information

Product Name:	ERK2/p38α MAPK-IN-1
Synonyms:	ERK2/p38α MAPK-IN-1
CAS:	1016427-72-7
MF:
MW:	0
EINECS:
Product Categories:
Mol File:	Mol File

ERK2/p38α MAPK-IN-1 Chemical Properties

Safety Information

MSDS Information

ERK2/p38α MAPK-IN-1 Usage And Synthesis

Uses

ERK2/p38α MAPK-IN-1 (Compound 1, In silico Hit-2) is a potent and selective ERK2 and p38α MAPK inhibitor, with an IC50 of 82 μM for ERK2. ERK2/p38α MAPK-IN-1 binds to the allosteric site of ERK2 and p38α MAPK in distinct manners. ERK2/p38α MAPK-IN-1 can be used for the research of type 2 diabetes[1].

References

[1] Hasegawa S, et al. Distinct binding modes of a benzothiazole derivative confer structural bases for increasing ERK2 or p38α MAPK selectivity. Biochem Biophys Res Commun. 2024 Apr 16;704:149707. DOI:10.1016/j.bbrc.2024.149707
[2] Kinoshita T, et al. Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assay. Bioorg Med Chem Lett. 2016 Feb 1;26(3):955-958. DOI:10.1016/j.bmcl.2015.12.056

ERK2/p38α MAPK-IN-1 Preparation Products And Raw materials

Tag:ERK2/p38α MAPK-IN-1(1016427-72-7) Related Product Information

HomePage | Member Companies | Advertising | Contact us | Previous WebSite | MSDS | CAS Index | CAS DataBase | Privacy | Terms | About Us
All products displayed on this website are only for non-medical purposes such as industrial applications or scientific research, and cannot be used for clinical diagnosis or treatment of humans or animals. They are not medicinal or edible.
According to relevant laws and regulations and the regulations of this website, units or individuals who purchase hazardous materials should obtain valid qualifications and qualification conditions.

ERK2/p38α MAPK-IN-1

Login

Fast registration