Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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Tel: |
821-50328103-801 18930552037 |
Email: |
3bsc@sina.com |
Products Intro: |
Product Name:NIDA 41020;N-(Piperidin-1-yl)-5-(4-Methoxyphenyl)-1-(2,4-dichlorophenyl)-4-Methyl-1H-pyrazole-3-carboxaMide CAS:502486-89-7 Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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Company Name: |
Sigma-Aldrich
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Tel: |
021-61415566 800-8193336 |
Email: |
orderCN@merckgroup.com |
Products Intro: |
Product Name:NIDA-41020 CAS:502486-89-7 Purity:>=97% (HPLC), solid Package:50MG Remarks:N8162-50MG
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Company Name: |
EMMX Biotechnology LLC
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Tel: |
888-539-0666 |
Email: |
info@emmx.com |
Products Intro: |
Product Name:NIDA 41020 CAS:502486-89-7 Purity:98% HPLC Package:5mg;10mg;25mg;50mg;100mg;250mg;500mg;1g
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| NIDA-41020 Basic information |
Product Name: | NIDA-41020 | Synonyms: | N-(Piperidin-1-yl)-5-(4-methoxyphenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide;1H-Pyrazole-3-carboxamide, 1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-4-methyl-N-1-piperidinyl-;NIDA-41020 >=97% (HPLC), solid;Alitretinoin Impurity 2 | CAS: | 502486-89-7 | MF: | C23H24Cl2N4O2 | MW: | 459.37 | EINECS: | | Product Categories: | | Mol File: | 502486-89-7.mol | |
| NIDA-41020 Chemical Properties |
storage temp. | 2-8°C | solubility | DMSO: ~16mg/mL | form | solid | color | off-white |
Hazard Codes | T | Risk Statements | 25-36/37/38 | Safety Statements | 26-45 | RIDADR | UN 2811 6.1 / PGIII | WGK Germany | 3 |
| NIDA-41020 Usage And Synthesis |
Uses | NIDA 41020 is an analog of rimonabant, which is a CB1 cannabinoic receptor antagonist that diminishes the behavioral effects of opiates and nicotine. | Biochem/physiol Actions | NIDA-41020 is a CB1 cannabinoid receptor antagonist. NIDA-41020 is structurally similar to Rimonabant, which is currently in clinical development. NIDA-41020 is less lipophilic; developed at NIDA as a potential radioligand for CB1 receptors, Ki = 4.1 nM [in comparison AM 251, AM 281, SR 141716 (Rimonabant) have Ki of 0.6, 4.5 and 1.8 nM respectively]. |
| NIDA-41020 Preparation Products And Raw materials |
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