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6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)-

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6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)- Suppliers list
Company Name: Hangzhou J&H Chemical Co., Ltd.  
Tel: 0571-+86-571-87396432
Email: sales@jhechem.com
Products Intro: Product Name:ET-JQ1-OH
CAS:2421153-77-5
Purity:98% HPLC Package:50KG;10KG;5KG;1KG
Company Name: Jilin Province Woda Biotechnology Co., Ltd.  
Tel: 13504435624
Email: 1927928688@qq.com
Products Intro: Product Name:ET-JQ1-OH
CAS:2421153-77-5
Purity:98%
Company Name: TargetMol Chemicals Inc.  
Tel: 4008200310
Email: marketing@tsbiochem.com
Products Intro: Product Name:ET-JQ1-OH
CAS:2421153-77-5
Purity:98% Package:100 mg；5 mg；50 mg
Company Name: Jiangsu Aikon Biopharmaceutical R&D Co.,Ltd.  
Tel: 025-66061636 18013972705
Email: qqyang@aikonchem.com
Products Intro: CAS:2421153-77-5
Purity:95% Package:1g;5g;10g
Company Name: Elucigen bio  
Tel: 13501719342
Email: wayne.zheng@elucigenbio.com
Products Intro: Product Name:(2R)-2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.02,]trideca-2(6),4,7,10,12-pentaen-9-yl]butanoic acid
CAS:2421153-77-5
Purity:97% LC/GC Package:10mg;25mg;50mg；100mg;250mg;500mg;1g;5g;10g Remarks:For research use only
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)- Basic information
Product Name:6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)-
Synonyms:6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)-;ET-JQ1-OH;(2R)-2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.02,?]trideca-2(6),4,7,10,12-pentaen-9-yl]butanoic acid
CAS:2421153-77-5
MF:C21H21ClN4O2S
MW:428.94
EINECS:
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Mol File:2421153-77-5.mol
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)- Structure
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)- Chemical Properties
Boiling point 663.8±65.0 °C(Predicted)
density 1.44±0.1 g/cm3(Predicted)
solubility Soluble to 100 mM in DMSO
pka4.11±0.10(Predicted)
Safety Information
MSDS Information
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)- Usage And Synthesis
Biological Activity(+)-JQ1 bump, acid functionalized is a BET bromodomain binding analog of (+)-JQ1 that selectively binds single point mutant form of Brd4 (Brd4BD2 L387A). Functionalized with a carboxylic acid group to enable onward chemistry. The position of the carboxylic acid group represents an 'exit vector' allowing modification without interfering with compound binding ability.
storageStore at -20°C
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)- Preparation Products And Raw materials
Tag:6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-α-ethyl-2,3,9-trimethyl-, (αR,6S)-(2421153-77-5) Related Product Information