基本信息
中文名称 | 4-[1-(Cyclohexyl-d11)-4-(4-fluorophenyl)-1H-iMidazol-5-yl]-2-pyriMidinaMine Dihydrochloride |
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中文同义词 | |
英文名称 | 4-[1-(Cyclohexyl-d11)-4-(4-fluorophenyl)-1H-iMidazol-5-yl]-2-pyriMidinaMine Dihydrochloride |
英文同义词 | 4-[1-(Cyclohexyl-d11)-4-(4-fluorophenyl)-1H-iMidazol-5-yl]-2-pyriMidinaMine Dihydrochloride;PF 670462-d11 |
CAS号 | |
分子式 | C19H11Cl2D11FN5 |
分子量 | 421.383662758 |
EINECS号 | |
相关类别 | |
Mol文件 | Mol File |
结构式 |
4-[1-(Cyclohexyl-d11)-4-(4-fluorophenyl)-1H-iMidazol-5-yl]-2-pyriMidinaMine Dihydrochloride 性质
用途
Labelled analogue of PF 670462, a potent and selective casein kinase 1ε (CK1ε) and CK1δ inhibitor. PF 670462 has been shown to inhibit PER protein nuclear translocation causing phase shifts in circadi an rhythms. PF 670462 attenuates methamphetamine-stimulated locomotion in vivo.