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| Product Name: | Mycro3 | | Synonyms: | Mycro3;ethyl 5-[[7-[chloro(difluoro)methyl]-5-(furan-2-yl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-1-phenylpyrazole-4-carboxylate;Mycro-3, >98%;1H-Pyrazole-4-carboxylic acid, 5-[[[7-(chlorodifluoromethyl)-5-(2-furanyl)pyrazolo[1,5-a]pyrimidin-2-yl]carbonyl]amino]-1-phenyl-, ethyl ester;Ethyl 5-(7-(chlorodifluoromethyl)-5-(furan-2-yl)pyrazolo[1,5-a]pyrimidine-2-carboxamido)-1-phenyl-1H-pyrazole-4-carboxylate;dimerization,Mycro 3,pancreatic,inhibit,adenocarcinoma,ductal,c-Myc,Inhibitor,PDA,Autophagy,Mycro3,MAX,Myc;ethyl 5-[7-(chlorodifluoromethyl)-5-(furan-2-yl)pyrazolo[1,5-a]pyrimidine-2-amido]-1-phenyl-1H-pyrazole-4-carboxylate | | CAS: | 944547-46-0 | | MF: | C24H17ClF2N6O4 | | MW: | 526.88 | | EINECS: | | | Product Categories: | | | Mol File: | 944547-46-0.mol |  |
| | Mycro3 Chemical Properties |
| density | 1.53±0.1 g/cm3(Predicted) | | storage temp. | Sealed in dry,Store in freezer, under -20°C | | solubility | DMSO : ≥ 100 mg/mL (189.80 mM) | | pka | 6.95±0.46(Predicted) | | form | Solid | | color | Light yellow to yellow |
| | Mycro3 Usage And Synthesis |
| Biological Activity | Mycro 3 is a potent selective Myc-Max dimerization inhibitor. It can be used in pancreatic cancer research. | | in vitro | Mycro 3 is a potent and selective c-Myc inhibitor in whole cell assays, with weak inhibitory activity against Activator protein 1 (AP-1). It has a superior specificity profile to its predecessors. It inhibits the interaction between c-Myc and Max. It has high selectivity and inhibits c-Myc/Max dimerization and conjugation with DNA. | | target | |
| | Mycro3 Preparation Products And Raw materials |
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